نتایج جستجو برای: angiogenic activity

تعداد نتایج: 1147308  

Journal: :Bioorganic & medicinal chemistry letters 2013
Sung Hee Hwang Aaron T Wecksler Guodong Zhang Christophe Morisseau Long V Nguyen Samuel H Fu Bruce D Hammock

To reduce the pro-angiogenic effects of sEH inhibition, a structure-activity relationship (SAR) study was performed by incorporating structural features of the anti-angiogenic multi-kinase inhibitor sorafenib into soluble epoxide hydrolase (sEH) inhibitors. The structural modifications of this series of molecules enabled the altering of selectivity towards the pro-angiogenic kinases C-RAF and v...

Journal: :Molecular cancer research : MCR 2014
Michael S Rogers Katherine Novak David Zurakowski Lorna M Cryan Anna Blois Eugene Lifshits Trond H Bø Anne M Oyan Elise R Bender Michael Lampa Soo-Young Kang Kamila Naxerova Karl-Henning Kalland Oddbjorn Straume Lars A Akslen Randolph S Watnick Judah Folkman George N Naumov

UNLABELLED The angiogenic switch, a rate-limiting step in tumor progression, has already occurred by the time most human tumors are detectable. However, despite significant study of the mechanisms controlling this switch, the kinetics and reversibility of the process have not been explored. The stability of the angiogenic phenotype was examined using an established human liposarcoma xenograft m...

Journal: :Journal of the American Academy of Dermatology 2009
Amy Nguyen Van Hoang Vivian Laquer Kristen M Kelly

UNLABELLED Angiogenesis is an important process in normal physiology and disease pathogenesis. Angiogenesis is controlled in a healthy body by a system of angiogenic growth factors and angiogenesis inhibitors. When angiogenic growth factors are predominantly expressed, blood vessel growth occurs and disease may result. Successful therapies have been developed that target growth factors, their r...

2015
Arianna Giacomini Sara Matarazzo Katiuscia Pagano Laura Ragona Sara Rezzola Michela Corsini Emanuela Di Salle Marco Presta Roberto Ronca

Fibroblast growth factor-8b (FGF8b) affects the epithelial/stromal compartments of steroid hormone-regulated tumors by exerting an autocrine activity on cancer cells and a paracrine pro-angiogenic function, thus contributing to tumor progression. The FGF8b/FGF receptor (FGFR) system may therefore represent a target for the treatment of steroid hormone-regulated tumors. The soluble pattern recog...

2015
Marie-Agnès Doucey Ioannis Xenarios

By merging computational systems modeling and experimental approaches, we have uncovered treatments reprogramming pro-angiogenic monocytes present in breast tumor into immunologically potent cells capable of mediating an anti-tumor immune response. The unraveled pathways and ligands which underlie monocyte pro-angiogenic activity have a strong predictive value for breast cancer patient relapse ...

Journal: :avicenna journal of phytomedicine 0
samaneh rahamoz haghighi department of plant breeding, faculty of new sciences and technologies, graduate university of advanced technology, kerman, iran malek hossein asadi department of biotechnology, institute of science and high technology and environmental sciences, graduate university of advanced technology, kerman, iran hassan akrami department of biology, faculty of basic science, razi university, kermanshah, iran amin baghizadeh department of biotechnology, institute of science and high technology and environmental sciences, graduate university of advanced technology, kerman, iran

objective: acorus calamus (a. calamus) has been used as a medicinal plant in asia for its effects on digestive system for the last 2000 years. to investigate the anti-cancer activity of rhizome of a. calamus, the ethanolic and methanolic extracts and essential oil of the rhizome were prepared and their effects were assessed on human gastric cancer cell line (ags). materials and methods: the via...

Journal: :Dalton transactions 2009
Raymond Wai-Yin Sun Miro Fei-Yeung Ng Ella Lai-Ming Wong Jingfei Zhang Stephen Sin-Yin Chui Lam Shek Tai-Chu Lau Chi-Ming Che

An oxo-bridged diruthenium(III) complex containing pyrazolato and pyrazole ligands is stable against ascorbic-acid reduction, induces apoptosis (60%, 48 h) against HeLa cells at 10 microM level and exhibits promising anti-angiogenic activity at its sub-cytotoxic concentrations. Other mononuclear ruthenium(III) complexes containing pyrazole ligands [Ru(pz)(4)X(2)](+) exhibit dual anti-angiogenic...

2014
Hao Ding Song Chen Wen-Qi Song You-Shui Gao Jun-Jie Guan Yang Wang Yuan Sun Chang-Qing Zhang

One of the big challenges in tissue engineering for treating large bone defects is to promote the angiogenesis of the tissue-engineered bone. Hypoxia inducible factor-1α (HIF-1α) plays an important role in angiogenesis-osteogenesis coupling during bone regeneration, and can activate a broad array of angiogenic factors. Dimethyloxaloylglycine (DMOG) can activate HIF-1α expression in cells at nor...

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