نتایج جستجو برای: binding mode

تعداد نتایج: 632612  

2012
Paweł Śledź Steffen Lang Christopher J Stubbs Chris Abell

Probing the pocket: A high-throughput fluorescence-based thermal shift (FTS) assay utilized different forms of a protein (in gray) to establish the binding mode of a ligand (see picture). The assay serves in the rapid evaluation of structure-activity binding-mode relationships for a series of ligands of Plk1, an important target of anticancer therapy.

2016
Katsuya Ohbuchi Yoshikazu Mori Kazuo Ogawa Eiji Warabi Masahiro Yamamoto Takatsugu Hirokawa

Transient receptor potential vanilloid type 1 (TRPV1) is a non-selective cation channel and a multimodal sensor protein. Since the precise structure of TRPV1 was obtained by electron cryo-microscopy, the binding mode of representative agonists such as capsaicin and resiniferatoxin (RTX) has been extensively characterized; however, detailed information on the binding mode of other vanilloids rem...

Journal: :Journal of Enzyme Inhibition and Medicinal Chemistry 2020

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