نتایج جستجو برای: carfilzomib

تعداد نتایج: 778  

Journal: :Blood 2012
David S Siegel Thomas Martin Michael Wang Ravi Vij Andrzej J Jakubowiak Sagar Lonial Suzanne Trudel Vishal Kukreti Nizar Bahlis Melissa Alsina Asher Chanan-Khan Francis Buadi Frederic J Reu George Somlo Jeffrey Zonder Kevin Song A Keith Stewart Edward Stadtmauer Lori Kunkel Sandra Wear Alvin F Wong Robert Z Orlowski Sundar Jagannath

Carfilzomib is a next-generation, selective proteasome inhibitor being evaluated for the treatment of relapsed and refractory multiple myeloma. In this open-label, single-arm phase 2 study (PX-171-003-A1), patients received single-agent carfilzomib 20 mg/m(2) intravenously twice weekly for 3 of 4 weeks in cycle 1, then 27 mg/m(2) for ≤ 12 cycles. The primary endpoint was overall response rate (...

Journal: :Blood 2015
Pieter Sonneveld Emilie Asselbergs Sonja Zweegman Bronno van der Holt Marie Jose Kersten Edo Vellenga Marinus van Marwijk-Kooy Annemiek Broyl Okke de Weerdt Sarah Lonergan Antonio Palumbo Henk Lokhorst

This multicenter phase 2 study of the European Myeloma Network investigated the combination of carfilzomib, thalidomide, and dexamethasone (KTd) as induction/consolidation therapy for transplant-eligible patients with previously untreated multiple myeloma (N = 91). During KTd induction therapy, patients received 4 cycles of carfilzomib 20/27 mg/m(2) (n = 50), 20/36 mg/m(2) (n = 20), 20/45 mg/m(...

2015
F Jonsson Y Ou L Claret D Siegel S Jagannath R Vij A Badros S Aggarwal R Bruno

Change in tumor size estimated using longitudinal tumor growth inhibition (TGI) modeling is an early predictive biomarker of clinical outcomes for multiple cancer types. We present the application of TGI modeling for subjects with multiple myeloma (MM). Longitudinal time course changes in M-protein data from relapsed and/or refractory MM subjects who received single-agent carfilzomib in phase I...

Journal: :The Lancet Oncology 2012

Journal: :Expert Opinion on Biological Therapy 2014

Journal: :Frontiers in Cell and Developmental Biology 2021

Despite several new therapeutic options, multiple myeloma (MM) patients experience relapses and inevitably become refractory to treatment. Insights into drug resistance mechanisms may lead the development of novel treatment strategies. The S100 family is comprised 21 calcium binding protein members with 17 genes located in 1q21 region, which commonly amplified MM. Dysregulated expression associ...

Journal: :American Journal of Hematology 2021

The MCRN-003/CCTGMYX.1 is a single arm phase II trial of weekly carfilzomib, cyclophosphamide and dexamethasone (wKCd), exploring convenient immunomodulator (IMiD)-free regimen in relapsed myeloma. Weekly carfilzomib (20/70 mg/m2), 40 mg 300 mg/m2 was delivered over 28-day cycles. primary endpoint overall response after four Secondary endpoints included toxicity, depth, PFS OS. Exploratory the ...

Journal: :The Journal of pharmacology and experimental therapeutics 2012
Sue Ellen Verbrugge Yehuda G Assaraf Ben A C Dijkmans George L Scheffer Marjon Al Debby den Uyl Ruud Oerlemans Elena T Chan Christopher J Kirk Godefridus J Peters Joost W van der Heijden Tanja D de Gruijl Rik J Scheper Gerrit Jansen

Bortezomib (BTZ), a registered proteasome inhibitor (PI) for multiple myeloma, has also been proposed as a potential antirheumatic agent. Its reported side effects, however, make it unappealing for long-term administration, and resistance may also develop. To overcome this, second-generation PIs became available. Here, we investigated whether a novel class of peptide epoxyketone-based PIs, incl...

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