نتایج جستجو برای: endothelin a receptor

تعداد نتایج: 13599043  

Journal: :International Journal of Human and Health Sciences (IJHHS) 2018

2012
Faquan Liang Suya Yang Lina Yao Luiz Belardinelli John Shryock

Endothelin receptor antagonists and phosphodiesterase type 5 inhibitors are used to treat pulmonary arterial hypertension. We tested the hypothesis that a selective endothelin type A receptor antagonist (ambrisentan) and a phosphodiesterase type 5 inhibitor (tadalafil) may act synergistically to relax endothelin-constricted pulmonary arteries. Rat isolated intrapulmonary arterial rings contract...

Journal: :The Journal of pharmacology and experimental therapeutics 2004
Mark C Kowala Natesan Murugesan John Tellew Kenneth Carlson Hossain Monshizadegan Carol Ryan Zhengxiang Gu Bridgette Kane Leena Fadnis Rose Ann Baska Sophie Beyer Susan Arthur Kenneth Dickinson Donglu Zhang Mark Perrone Pam Ferrer Mary Giancarli Jergen Baumann Eileen Bird Balkrushna Panchal Yifan Yang Nick Trippodo Joel Barrish John E Macor

Angiotensin II and endothelin-1 activate their respective AT(1) and ET(A) receptors on vascular smooth muscle cells, producing vasoconstriction, and both peptides are implicated in the pathogenesis of essential hypertension. Angiotensin II potentiates the production of endothelin, and conversely endothelin augments the synthesis of angiotensin II. Both AT(1) and ET(A) receptor antagonists lower...

Objectives: Endothelin-1 is a strong constrictor of blood vessels that is secreted by endothelial cells and identified as the strongest vascular constrictor. The aim of the present study was to investigate the effect of eight week aerobic exercise on the endothelin-1 concentration of plasma and its relationship with blood pressure in elderly postmenopausal women. Methods & Materials: A to...

1998
Mario Zuccarello Riccardo Boccaletti Alberto Romano Robert M. Rapoport

Cerebral Vasospasm Induced − Endothelin B Receptor Antagonists Attenuate Subarachnoid Hemorrhage Print ISSN: 0039-2499. Online ISSN: 1524-4628 Copyright © 1998 American Heart Association, Inc. All rights reserved. is published by the American Heart Association, 7272 Greenville Avenue, Dallas, TX 75231 Stroke doi: 10.1161/01.STR.29.9.1924 1998;29:1924-1929 Stroke. http://stroke.ahajournals.org/c...

2012
Daddam Jayasimha Rayalu Chandrabose Selvaraj Sanjeev Kumar Singh Ramakrishan Ganeshan Nagapatla Udaya Kumar Panthangi Seshapani

In cardiovascular system, activation of Endothelin receptors causes vasoconstriction which leads to Pulmonary Arterial Hypertension (PAH). Endothelin receptor antagonism has emerged as an important therapeutic strategy in pulmonary arterial hypertension. Bosentan is intended to affect vasoconstriction, hypertrophic and fibrotic effects by blocking the actions of receptors ET(A) and ET(B). In th...

Journal: :Cancer research 1999
A Bagnato D Salani V Di Castro J R Wu-Wong R Tecce M R Nicotra A Venuti P G Natali

In the present study, we have investigated the expression of endothelin 1 (ET-1) and the ET(A) receptor (ET(A)R) and ET(B) receptor (ET(B)R) in primary (n = 30) and metastatic (n = 8) ovarian carcinomas and their involvement in tumor growth. By reverse transcription-PCR and Northern blot analysis, we detected ET-1 mRNA in 90% of primary and 100% of metastatic ovarian carcinomas. ET-1 mRNA expre...

Journal: :Circulation 2001
A Seed J McMurray

tables or figures and should relate solely to an article published in Circulation within the preceding 12 weeks. Authors of letters selected for publication will receive prepublication proofs, and authors of the article cited in the letter will be invited to reply. Replies must be signed by all authors listed in the original publication. Please submit three typewritten, double-spaced copies of ...

Journal: :Pharmacological reports : PR 2012
Aleksandra Piechota-Polańczyk Anna Gorąca

BACKGROUND The potent vasoconstrictor endothelin-1 has been implicated in the pathogenesis of plasma oxidative stress seen in sepsis. The selective endothelin receptor blockers BQ123 and BQ788 were used to investigate the importance of selective endothelin receptor blockage in modulating oxidative stress during endotoxemia. METHODS The study was performed on male Wistar rats (n = 6 per group)...

Journal: :American journal of physiology. Heart and circulatory physiology 2008
David B Murray Jason D Gardner Gregory L Brower Joseph S Janicki

The objective of this study was to investigate the effect a nonselective endothelin-1 (ET-1) receptor antagonist (bosentan) had on the acute myocardial remodeling process including left ventricular (LV) mast cells and matrix metalloproteinase (MMP) activity secondary to volume overload. Additionally, we investigated the overall functional outcome of preventative endothelin receptor antagonism d...

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