نتایج جستجو برای: acetylcholinesterase inhibitor

تعداد نتایج: 217751  

Journal: :Pest management science 2010
Lihua Wang Yueliang Zhang Zhaojun Han Yanhe Liu Jichao Fang

BACKGROUND Laodelphax striatellus (Fallén) is a major pest of cultivated rice and is commonly controlled in China with the organophosphate insecticides. To develop a better resistance management strategy, a chlorpyrifos-resistant strain of L. striatellus was selected in the laboratory, and its cross-resistance to other insecticides and possible mechanisms of the chlorpyrifos resistance were inv...

2012
Zhenxin Zhang Lu Yu Maren Gaudig Barbara Schäuble Ute Richarz

BACKGROUND Acetylcholinesterase inhibitors are considered standard of care for Alzheimer's disease in many countries. Galantamine is an acetylcholinesterase inhibitor that may also act via allosteric modulation of nicotinic acetylcholine receptors. Therefore, it may provide benefits compared with other acetylcholinesterase inhibitors. The present study compared galantamine (n = 116) with donepe...

2018
Matheus Thomaz Nogueira Silva Lima Larissa Batista dos Santos Rafael Wesley Bastos Jacques Robert Nicoli Jacqueline Aparecida Takahashi

Major health challenges as the increasing number of cases of infections by antibiotic multiresistant microorganisms and cases of Alzheimer's disease have led to searching new control drugs. The present study aims to verify a new way of obtaining bioactive extracts from filamentous fungi with potential antimicrobial and acetylcholinesterase inhibitory activities, using epigenetic modulation to p...

Journal: :Molecules 2016
Michalina Hebda Marek Bajda Anna Więckowska Natalia Szałaj Anna Pasieka Dawid Panek Justyna Godyń Tomasz Wichur Damijan Knez Stanislav Gobec Barbara Malawska

Cholinesterases and amyloid beta are one of the major biological targets in the search for a new and efficacious treatment of Alzheimer's disease. The study describes synthesis and pharmacological evaluation of new compounds designed as dual binding site acetylcholinesterase inhibitors. Among the synthesized compounds, two deserve special attention--compounds 42 and 13. The former is a sacchari...

2016
Woosuk Kim Hee Sun Yim Dae Young Yoo Hyo Young Jung Jong Whi Kim Jung Hoon Choi Yeo Sung Yoon Dae Won Kim In Koo Hwang

BACKGROUND Cadmium leads to learning and memory impairment. Dendropanax morbifera Léveille stem extract (DMS) reduces cadmium-induced oxidative stress in the hippocampus. We investigated the effects of DMS on cadmium-induced impairments in memory in rats. METHODS Cadmium (2 mg/kg), with or without DMS (100 mg/kg), was orally administered to 7-week-old Sprague-Dawley rats for 28 days. Galantam...

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