نتایج جستجو برای: oral dosing

تعداد نتایج: 277969  

Journal: :Cancer research 2000
S R Wedge D J Ogilvie M Dukes J Kendrew J O Curwen L F Hennequin A P Thomas E S Stokes B Curry G H Richmond P F Wadsworth

There is evidence that vascular endothelial growth factor (VEGF) contributes to solid tumor growth through the promotion of both angiogenesis and tumor vascular permeability. To abrogate VEGF signaling, we developed a small molecular weight inhibitor of VEGF receptor tyrosine kinase (RTK) activity that was compatible with chronic oral administration. ZD4190, a substituted 4-anilinoquinazoline, ...

Journal: :Therapeutics and Clinical Risk Management 2006
Frieder Bauss Ralph C Schimmer

Osteoporosis is a major healthcare problem that continues growing as the population ages. Sufferers become increasingly susceptible to fractures, which compromise physical and emotional health and increase healthcare costs. Bisphosphonates are the most widely used medicines for the treatment and prevention of postmenopausal osteoporosis. However, therapeutic adherence is suboptimal, meaning tha...

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2005
Eyal Sobol Boris Yagen Ilan Winkler Malka Britzi Dan Gibson Meir Bialer

The pharmacokinetics and metabolism of 2,2,3,3-tetramethylcyclopropanecarbonylurea (TMCU), a potent anticonvulsant compound, were studied in male Sprague-Dawley rats following i.v. (5 mg/kg), oral (20 mg/kg), and i.p. (20 mg/kg) administrations. Urine samples were analyzed by gas chromatography-mass spectrometry (GC/MS) and liquid chromatography-mass spectrometry. Plasma samples were analyzed b...

2015
James V. Cassella Daniel A. Spyker Paul P. Yeung

OBJECTIVE This randomized, double-blind, active- and placebo-controlled, crossover, thorough QT study assessed the effect of two inhaled loxapine doses on cardiac repolarization as measured by corrected QT (QTc) interval in healthy subjects (ClinicalTrials.gov NCT01854710). METHODS Subjects received two doses of inhaled loxapine (10 mg) 2 hours apart+oral placebo, two doses of inhaled placebo...

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