Pyrazolines are biologically and pharmaceutically very active scaffolds. Derivatives of. (3,5-diphenyl-4,5-dihydro-1H-pyrazol-1-yl)(phenyl)methanone were synthesized by the cyclization of chalcones (1a-c) with substituted benzyl hydrazides (2a-e) using a few drops of piperidine as catalyst. Structures of all the synthesized compounds were confirmed by FTIR, 1H NMR, 13C NMR and mass spectrometri...

Broomrape weeds (Orobanche and Phelipanche spp.) are noxious parasites that infect crops using haustoria formed at the tip of their radicles. Dichloromethane extract obtained from roots Convolvulus arvensis strongly inhibits radicle growth broomrape weeds. A complex mixture arvensic acids was isolated as metabolites responsible inhibitory activity C. against via activity-guided fractionation 1H...

Fractions obtained from partitioning of aerial methanolic extract of Euphorbia Aelleniiwith chloroform (E2), ethyl acetate (E3), n-butanol (E4) and water (E5) were investigated in vitro for their phytotoxicity, insecticidal, anti-leishmanial, cytotoxicity, antibacterial and antifungal activities. Sample E2 appeared to have significant phytotoxic activity. In the insecticidal screening study onl...

Bioassay-directed fractionation of a CH(2)Cl(2)-MeOH (1:1) extract of the aerial parts of Flourensia cernua led to the isolation of three phytotoxic compounds, namely, dehydroflourensic acid (1), flourensadiol (2) and methyl orsellinate (3). Dehydroflourensic acid is a new natural product whose structure was established by spectral means. In addition, the known flavonoid ermanin and seven hithe...

The polyether antibiotic maduramicin and its methyl ester derivative inhibited photophosphorylation and proton uptake in isolated spinach chloroplasts. Both compounds also enhanced basal and phosphorylating electron transport and stimulated Mg(2+)-dependent ATPase activity, therefore, they behave as uncouplers of photophosphorylation being the methyl ester derivative more potent than the parent...

Twelve essential oils from Mediterranean aromatic plants were tested for their phytotoxic activity, at different doses, against the germination and the initial radicle growth of seeds of Raphanus sativus, Lactuca sativa and Lepidium sativum. The essential oils were obtained from Hyssopus officinalis, Lavandula angustifolia, Majorana hortensis, Melissa officinalis, Ocimum basilicum, Origanum vul...

Nitrodiphenylethers, Energy-Transfer Inhibition of ATP Synthesis, Herbicides, Photosynthetic Electron Transport, Pigment Bleaching Nitrodiphenylethers substituted with Cl, CF3, and other comparatively simple substituents are compared with respect to their primary effects on the photosynthetic apparatus. These are direct electron-transport inhibition, energy-transfer inhibition (of ATP synthesis...