نتایج جستجو برای: pik3ca

تعداد نتایج: 2433  

2018
Hua Li Shubo Chen Hui Li Jianxin Cui Yunhe Gao Dianchao Wu Shangfeng Luan Yan Qin Tongshan Zhai Dengxiang Liu Zhibin Huo

Background Increasing evidence suggests that dysregulation of phosphatidylinositol-4, 5-bisphosphate 3-kinase, catalytic subunit alpha (PIK3CA) plays an important role in carcinogenesis. However, the relationship between PIK3CA expression and gastric cancer (GC) prognosis remains controversial. Methods We searchedPubMed, Embase, Web of Science, and the Cochrane Library databases for relevant ...

Journal: :Oncology reports 2007
Irina Fenic Klaus Steger Christin Gruber Christoph Arens Joachim Woenckhaus

PIK3CA, which encodes the catalytic subunit, p110-alpha, of phosphatidylinositol 3-kinase (PI3K), is implicated in the development and progression of numerous neoplasias including head and neck squamous cell carcinoma (HNSCC). In the present study, we investigated the occurrence of PIK3CA hot-spot mutations in exons 9 and 20, the genomic gain and amplification of PIK3CA, the expression of PIK3C...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2007
Gizeh Pérez-Tenorio Liza Alkhori Birgit Olsson Marie Ahnström Waltersson Bo Nordenskjöld Lars Erik Rutqvist Lambert Skoog Olle Stål

PURPOSE The phosphatidylinositol 3'-kinase/Akt pathway is frequently altered in breast cancer. PTEN, a phosphatase that opposes the effect of phosphatidylinositol 3'-kinase, can be mutated or lost, whereas the PIK3CA gene is mutated. These have been proposed as alternative mechanisms, and their clinicalpathology significance is under discussion. In this study, we aimed to explore whether PIK3CA...

2017
Jean-François Laes Sebastien Sauvage Gregori Ghitti

The mechanistic target of the rapamycin (mTOR) pathway is frequently activated in human cancers. Our objective was to evaluate relationships between mTOR-pathway activity and functional mutations in the upstream genes PIK3CA and PTEN in solid-tumor biopsies from a broad selection of cancer types. Formalin-fixed paraffin-embedded (FFPE) tumor samples were analyzed by immunohistochemistry (IHC) a...

Journal: :Molecular cancer therapeutics 2007
Jing Wang Karen Kuropatwinski Jennie Hauser Michael R Rossi Yunfei Zhou Alexis Conway Julie L C Kan Neil W Gibson James K V Willson John K Cowell Michael G Brattain

PIK3CA, encoding the p110alpha catalytic subunit of phosphatidylinositol 3-kinase (PI3K), is mutated in a variety of human cancers. We screened the colon cancer cell lines previously established in our laboratory for PIK3CA mutations and found that four of them harbored gain of function mutations. We have now compared a panel of mutant and wild-type cell lines for cell proliferation and surviva...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2013
Fiona L Day Robert N Jorissen Lara Lipton Dmitri Mouradov Anuratha Sakthianandeswaren Michael Christie Shan Li Cary Tsui Jeannie Tie Jayesh Desai Zheng-Zhou Xu Peter Molloy Vicki Whitehall Barbara A Leggett Ian T Jones Stephen McLaughlin Robyn L Ward Nicholas J Hawkins Andrew R Ruszkiewicz James Moore Dana Busam Qi Zhao Robert L Strausberg Peter Gibbs Oliver M Sieber

PURPOSE PIK3CA and PTEN mutations are prevalent in colorectal cancer and potential markers of response to mitogen-activated protein/extracellular signal-regulated kinase inhibitors and anti-EGF receptor antibody therapy. Relationships between phosphoinositide 3-kinase (PI3K) pathway mutation, clinicopathologic characteristics, molecular features, and prognosis remain controversial. EXPERIMENT...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2016
Sibylle Loibl Silvia Darb-Esfahani Jens Huober Alexander Klimowicz Jenny Furlanetto Bianca Lederer Arndt Hartmann Holger Eidtmann Berit Pfitzner Peter A Fasching Katharina Tiemann Christian Jackisch Keyur Mehta Gunter von Minckwitz Michael Untch Carsten Denkert

BACKGROUND The PI3K/AKT pathway and phosphatase and tensin homolog (PTEN) aberrations are common in breast cancer. We investigated the correlation between phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha (PIK3CA), PTEN, p4EBP1 (phosphorylated E4 binding protein 1), and pathologic complete response (pCR) in patients receiving neoadjuvant therapy. EXPERIMENTAL DESIGN We re...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2006
Frank Schönleben Wanglong Qiu Nancy T Ciau Daniel J Ho Xiaojun Li John D Allendorf Helen E Remotti Gloria H Su

PURPOSE Recent studies have reported high frequencies of somatic mutations in the phosphoinositide-3-kinase catalytic-alpha (PIK3CA) gene in various human solid tumors. More than 75% of those somatic mutations are clustered in the helical (exon 9) and kinase domains (exon 20). The three hot-spot mutations, E542K, E545K, and H1047R, have been proven to elevate the lipid kinase activity of PIK3CA...

2012
Craig P. Carden Adam Stewart Parames Thavasu Emma Kipps Lorna Pope Mateus Crespo Susana Miranda Gerhardt Attard Michelle D. Garrett Paul A. Clarke Paul Workman Johann S. de Bono Martin Gore Stan B Kaye Udai Banerji

Evidence that the phosphoinositide 3-kinase (PI3K) pathway is deregulated in ovarian cancer is largely based on the analysis of surgical specimens sampled at diagnosis and may not reflect the biology of advanced ovarian cancer. We aimed to investigate PI3K signaling in cancer cells isolated from patients with advanced ovarian cancer.Ascites sampleswere analyzed from88patients, ofwhom61 received...

پایان نامه :وزارت علوم، تحقیقات و فناوری - دانشگاه اراک - دانشکده علوم پایه 1393

فسفاتیدیل اینوزیتول 3- کینازها (pi3ks) گروهی از لیپید کینازهای مسیرهای انتقال پیام هستند که در تنظیم فرایندهای تکثیر، چسبندگی، بقا و تحرک سلولی مشارکت دارند. کلاس iاین خانواده آنزیمی از دو زیر واحد کاتالیتیکی و تنظیمی تشکیل شده است. جهش های زیر واحد کاتالیتیکی که توسط ژن pik3caکد می شود، موجب افزایش فعالیت آنزیم و رشد کنترل نشده سلول ها می شوند. مطالعات گذشته درصد بالایی از جهش های این ژن را در...

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