نتایج جستجو برای: substituent effects

تعداد نتایج: 1548409  

Journal: :The Journal of pharmacology and experimental therapeutics 2012
Jenny L Wiley Dana E Selley Pinglang Wang Rudresha Kottani Srinivas Gadthula Anu Mahadeven

The prototypic cannabinoid type 1 (CB₁) receptor antagonist/inverse agonist, rimonabant, is comprised of a pyrazole core surrounded by a carboxyamide with terminal piperidine group (3-substituent), a 2,4-dichlorophenyl group (1-substituent), a 4-chlorophenyl group (5-substituent), and a methyl group (4-substituent). Previous structure-activity relationship (SAR) analysis has suggested that the ...

Journal: :The Journal of organic chemistry 2006
Lauri Toom Agnes Kütt Ivari Kaljurand Ivo Leito Henrik Ottosson Helena Grennberg Adolf Gogoll

Basicity constants for a series of 3,7-diazabicyclo[3.3.1]nonane derivatives in acetonitrile with a variation over 13 orders of magnitude have been determined using a spectrophotometric titration technique. An excellent correlation between basicity and calculated proton affinities obtained at PCM-B3LYP/6-31+G(d)//B3LYP/6-31G(d) level was found. The results are discussed in terms of substituent ...

2001
KEVIN C. GROSS PAUL G. SEYBOLD

Substituent effects on the physical properties and pKa of phenol were studied using density functional theory [B3LYP /6-311G(d,p)] calculations. Substituents alter the physical properties of phenol such as the hydroxyl-group C-0 and 0-H bond lengths, the C-0-H bond angle, and the energy barrier to rotation about the C-0 bond, and also influence the hydroxyl-group pK •. Except for the rotational...

Journal: :Bulletin of the Chemical Society of Japan 1990

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