نتایج جستجو برای: thiazolidin 4 one

تعداد نتایج: 3010807  

Journal: :Acta Crystallographica Section E Structure Reports Online 2013

2016
Barbaros Eroglu Keriman Ozadali-Sari Oya Unsal-Tan Sriram Dharmarajan Perumal Yogeeswari Ayla Balkan

To develop novel antimycobacterial agents, a new series of thiazolidinone-azole hybrids 4a-b, 5a-b and 6-13 were designed and synthesized. Thiazolidin-4-ones (4a-b and 5a-b) were obtained by the reaction of Schiff bases and hydrazones (2a-b and 3a-b) with mercaptoacetic acid. 5-Benzylidene derivatives (6-13) were gained by treatment of 5a-b with appropriate benzaldehydes according to Knoevenage...

Journal: :Bioorganic & medicinal chemistry letters 2012
Hua Chen Tianyu Yang Sinan Wei Hongzhi Zhang Rui Li Zhanbin Qin Xiaoliu Li

Novel bicyclic iminosugar derivatives fused thiazolidin-4-one were conveniently synthesized by double Pummerer rearrangements, and their HIV reverse transcriptase (RT) inhibitory activities were preliminary examined. The notable anti-HIV-RT activity demonstrated that such bicyclic azasugars hold potential as a new kind of HIV-RT inhibitors.

Journal: :Beilstein Journal of Organic Chemistry 2008
Deepa Pandey Wahajul Haq Seturam B Katti

In search of new erythromycin derivatives 3-O-[gamma-(4-oxo-2-aryl-thiazolidin-3-yl)butyryl]erythromycin A derivatives have been synthesized. The 3-hydroxy group was derivatised to a primary amine and subsequently the thiazolidinone nucleus was generated at the amino functionality through DCC mediated one-pot three-component reaction in good yields.

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید