نتایج جستجو برای: brafv600e

تعداد نتایج: 835  

Journal: :View 2023

The back cover image describes a DCNN model based on ultrasound images to predict the BRAFV600E mutation in thyroid nodules which achieved encouraging predictive performance test sets from four hospitals (AUC 0.84–0.93). This might provide non-invasive and convenient method for predicting assist clinicians select more appropriate management patients with or cancer.

2016
Michaël Cerezo Stéphane Rocchi

Melanoma is the most lethal form of skin cancer. Until 2011, the favored therapy was chemotherapy despite their low efficiency. Spectacular progresses were made in melanoma treatment using targeted therapies anti-BRAFV600E / anti-MEK and immunotherapy antiCTLA-4 / anti PD-1. Unfortunately, more than 50% of patients present intrinsic or acquire resistance and are in treatment failure. So identif...

Journal: :Annals of Oncology 2022

Current knowledge on biomarkers (BRAFV600E/RAS mutations) is mainly based metastatic colorectal cancer (mCRC) patients with proficient mismatch repair (pMMR) tumors. It uncertain whether these have the same implications in deficient (dMMR) mCRC patients. Our aim to provide insight value of Lynch syndrome, BRAFV600E and RAS mutation status treatment regimens survival dMMR treated outside clinica...

Journal: :British Journal of Surgery 2022

Abstract Background NHS England’s reorganization of genomic testing has provided an opportunity to explore molecular as part thyroid nodule diagnostics and the routine postoperative histology. Aim Routine in service not previously been explored. This study aims evaluate whether (1) there is sufficient material perform this on FNAC cytologically indeterminate nodules (2) what yield from (3) post...

Journal: :European Journal of Medicinal Chemistry 2021

The synergistic effect of dual inhibition serine/threonine protein kinases that are involved in the same signalling pathway diseases can exert superior biological benefits for treatment these diseases. In present work, a new series (imidazol-5-yl)pyrimidine was designed and synthesized as inhibitors BRAFV600E p38? which considered key regulators mitogen-activated kinase (MAPK) pathway. target c...

2015
Brian J. Capaldo Devin Roller Mark J. Axelrod Alex F. Koeppel Emanuel F. Petricoin Craig L. Slingluff Michael J. Weber Aaron J. Mackey Daniel Gioeli Stefan Bekiranov Keiran Smalley

Fifty percent of cutaneous melanomas are driven by activated BRAFV600E, but tumors treated with RAF inhibitors, even when they respond dramatically, rapidly adapt and develop resistance. Thus, there is a pressing need to identify the major mechanisms of intrinsic and adaptive resistance and develop drug combinations that target these resistance mechanisms. In a combinatorial drug screen on a pa...

2014
Pierre Vanden Borre Viswanath Gunda David G. McFadden Peter M. Sadow Shohreh Varmeh Maria Bernasconi Sareh Parangi

Anaplastic (ATC) and refractory papillary thyroid cancer (PTC) lack effective treatments. Inhibition of either oncogenic BRAF or SRC has marked anti-tumor effects in mouse models of thyroid cancer, however, neither drug induces notable apoptosis. Here we report that the SRC-inhibitor dasatinib further sensitizes BRAFV600E-positive thyroid cancer cells to the BRAFV600E-inhibitor PLX4720. Combine...

Journal: :Blood 2014
Rikhia Chakraborty Oliver A Hampton Xiaoyun Shen Stephen J Simko Albert Shih Harshal Abhyankar Karen Phaik Har Lim Kyle R Covington Lisa Trevino Ninad Dewal Donna M Muzny Harshavardhan Doddapaneni Jianhong Hu Linghua Wang Philip J Lupo M John Hicks Diana L Bonilla Karen C Dwyer Marie-Luise Berres Poulikos I Poulikakos Miriam Merad Kenneth L McClain David A Wheeler Carl E Allen D Williams Parsons

Langerhans cell histiocytosis (LCH) is a myeloproliferative disorder characterized by lesions composed of pathological CD207(+) dendritic cells with an inflammatory infiltrate. BRAFV600E remains the only recurrent mutation reported in LCH. In order to evaluate the spectrum of somatic mutations in LCH, whole exome sequencing was performed on matched LCH and normal tissue samples obtained from 41...

Journal: :Integrative biology : quantitative biosciences from nano to macro 2014
Ling Yu Li Xia Gao Xiao Qing Ma Fang Xin Hu Chang Ming Li Zhisong Lu

The BRAF(V600E) inhibitor PLX4032 (Vemurafenib) is an FDA-approved new drug for the treatment of metastatic melanomas, which specifically inhibits the RAS/MEK/ERK signaling pathway to control cell proliferation and adhesion. However, no study has been carried out to investigate the role of intracellular oxidative balance in PLX4032-induced tumor growth inhibition. Herein, for the first time, su...

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