نتایج جستجو برای: hek293

تعداد نتایج: 3784  

2013
Martin J. Gunthorpe Sara Luis Hannan Darren Smart

SB-705498 is a potent, selective and orally bioavailable transient receptor potential vanilloid 1 (TRPV1) receptor antagonist with a pIC50 of 7.1. SB-705498 potently inhibits capsaicin-induced activation of human TRPV1 expressed in 1321N1 cells or HEK293 cells with apparent pKi of 7.5 or 7.6, respectively. Coapplication of 100 nM SB-705498 rapidly, completely and reversibly inhibits hTRPV1 expr...

Journal: :Food Science and Technology 2022

Cancer is a disease that invades the lives of millions people each year. Chemotherapy currently most effective treatment however resulting in many adverse effects to human body. Alternative treatments are being explored overcome this obstacle. Peptides possess radical scavenging activity and bioactive properties can be advantageous prevention chronic diseases. In study, Lablab purpureus isolate...

Journal: :Molecules 2014
Fang Xu Hong Chen Xuelan He Jingyi Xu Bingbing Xu Biyun Huang Xue Liang Mu Yuan

α1-Adrenoceptors (ARs; 1A, 1B, and 1D) have been determined to perform different prominent functions in the physiological responses of the sympathetic nervous system. A high-throughput screening assay (HTS) was set up to detect α1-AR subtype-selective agonists by a dual-luciferase reporter assay in HEK293 cells. Using the HTS assay, two novel compounds, CHE3 and CHK3, were discovered as α1-ARs ...

2015
Borja Díaz de Greñu José García-Calvo José Cuevas Gabriel García-Herbosa Begoña García Natalia Busto Saturnino Ibeas Tomás Torroba Blanca Torroba Antonio Herrera Sebastian Pons

Selected new fluorogenic probes that interact in different ways with Hg and MeHg have been prepared and used for the chemical speciation of both cations in aqueous solution as well as in HEK293 cells. The best selective speciation of Hg and MeHg has been achieved by in vitro approaches based on fluorogenic probes supported in cultured cells, due to the particular sensitivity of the HEK293 cells...

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