نتایج جستجو برای: xenobiotic metabolizing

تعداد نتایج: 9468  

2015
Wafa Hassen Alboukadel Kassambara Thierry Reme Surinder Sahota Anja Seckinger Laure Vincent Guillaume Cartron Jérôme Moreaux Dirk Hose Bernard Klein

Resistance to chemotherapy is a major limitation of cancer treatments with several molecular mechanisms involved, in particular altered local drug metabolism and detoxification process. The role of drug metabolism and clearance system has not been satisfactorily investigated in Multiple Myeloma (MM), a malignant plasma cell cancer for which a majority of patients escapes treatment. The expressi...

Journal: :Molecular pharmacology 2004
Ibtissam Echchgadda Chung S Song Arun K Roy Bandana Chatterjee

Dehydroepiandrosterone sulfotransferase (SULT2A1) is a cytosolic enzyme that mediates sulfo-conjugation of endogenous hydroxysteroids (dehydroepiandrosterone, testosterone, bile acids), and diverse xenobiotic compounds. Upon sulfonation, SULT2A1 substrates become polar and water-soluble and thus suitable for rapid excretion. SULT2A1 is abundantly expressed in the liver and intestine. Recent evi...

2006
Thomas Thum Veit J. Erpenbeck Julia Moeller Jens M. Hohlfeld Norbert Krug Jürgen Borlak

BACKGROUND Cytochrome P450 monooxygenases (CYP) play an important role in the defense against inhaled toxicants, and expression of CYP enzymes may differ among various lung cells and tissue compartments. METHODS We studied the effects of tobacco smoke in volunteers and investigated gene expression of 19 CYPs and 3 flavin-containing monooxygenases, as well as isoforms of glutathione S-transfer...

Journal: :The Journal of pharmacology and experimental therapeutics 2008
Connie Cheung Frank J Gonzalez

Cytochrome P450s (P450s) are important enzymes involved in the metabolism of xenobiotics, particularly clinically used drugs, and are also responsible for metabolic activation of chemical carcinogens and toxins. Many xenobiotics can activate nuclear receptors that in turn induce the expression of genes encoding xenobiotic metabolizing enzymes and drug transporters. Marked species differences in...

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