نتایج جستجو برای: ccufe2o4sio2c3 pyrazole c4so3 h2pw

تعداد نتایج: 3198  

The physical and chemical properties of Pyrazole and Pyrazoline molecules were theoreticallystudied by Gaussian 03, software with NMR and Molecular orbital calculations at B3LYP/6-31G andB3LYP/6-31+G(d) levels, in gas phase and solution. In this study a comparison effect of threesolvents with different dielectric constants on Pyrazole and Pyrazoline molecules in aspect energyinteraction between...

Journal: :European Journal of Chemistry 2022

In-silico quantitative structure-activity relationship (QSAR) study was performed to develop a model on series of novel pyrazole derivatives containing acetamide moiety which exhibited considerable antiproliferative activity against human colorectal adenocarcinoma cell line HT-29. The obtained has correlation coefficient (r) 0.9693, squared (r2) 0.9395 and leave-one-out (LOO) cross-validation (...

Journal: :Berichte der deutschen chemischen Gesellschaft 1904

2010
Guiqiu Yang Hongcai Xu Huibin Yang Haibo Yu

The pyazole ring in the title compound, C(6)H(9)ClN(2), is almost planar (r.m.s. deviation = 0.003 Å). In the crystal, mol-ecules are linked by C-H⋯N inter-actions, forming [100] chains.

Journal: :Journal of Materials Chemistry C 2021

In this contribution pyrazole is identified as an excellent anchor group that forms high quality films under pH controlled conditions, allowing the modulation of electrical properties with a more efficient electronic coupling in basic conditions.

2015
Gregory M. Ferrence Joshua L. Kocher

The title compound, C7H14N2Si, crystallizes in a tetra-gonal space group and exists as an N-H⋯N hydrogen-bonded tetra-mer, formed around the crystallographic fourfold rotoinversion axis. The mol-ecular identity is clearly the 5-tri-methyl-silyl-3-methyl-1H-pyrazole tautomer and the structure is isomorphous with that of 5-tert-butyl-3-methyl-1H-pyrazole [Foces-Foces & Trofimenko (2001 ▶). Acta C...

Journal: :Organic letters 2011
Rahul Kumar Irishi N N Namboothiri

A base mediated reaction of α-diazo-β-ketosulfone with nitroalkenes affords sulfonylpyrazoles as single regioisomers in excellent yield in a one-pot room temperature reaction. Aryl, heteroaryl, styrenyl, alkyl, hydroxymethyl, and hydrazinyl groups could be introduced on the pyrazole ring by the appropriate choice of nitroalkenes. Synthesis of sulfonylpyrazole fused to other heterocycles and app...

2014
B. Narayana Vinutha V. Salian Balladka K. Sarojini Jerry P. Jasinski

In the title compound, C22H25ClN2O, the pyrazole ring exhibits an envelope conformation with the methine C atom as the flap. The benzene rings are twisted by 3.3 (5) and 84.6 (5)° from the pyrazole mean plane, and are inclined to each other by 81.4 (4)°. In the crystal, pairs of weak C-H⋯O hydrogen bonds form centrosymmetric dimers with an R 2 (2)(16) graph-set motif. C-H⋯π inter-actions link t...

2014
Karikere Ekanna Manoj Kumar Parameshwar Adimoole Suchetan Bandrehalli Siddagangaiah Palakshamurthy Shankar Madan Kumar Neratur Krishnappagowda Lokanath Swamy Sreenivasa

In the title compound, C16H8F6N2, the dihedral angle between the pyrazole and di-fluoro-benzene rings is 50.30 (13)°, while those between the pyrazole and fluoro-benzene rings and between the di-fluoro-benzene and fluoro-benzene rings are 38.56 (13) and 53.50 (11)°, respectively. Aromatic π-π stacking inter-actions between adjacent di-fluoro-benzene rings [centroid-centroid separation = 3.6082 ...

Journal: :Journal of medicinal chemistry 2015
Zachary Miller Keun-Sik Kim Do-Min Lee Vinod Kasam Si Eun Baek Kwang Hyun Lee Yan-Yan Zhang Lin Ao Kimberly Carmony Na-Ra Lee Shou Zhou Qingquan Zhao Yujin Jang Hyun-Young Jeong Chang-Guo Zhan Wooin Lee Dong-Eun Kim Kyung Bo Kim

We performed a virtual screen of ∼340 000 small molecules against the active site of proteasomes followed by in vitro assays and subsequent optimization, yielding a proteasome inhibitor with pyrazole scaffold. The pyrazole-scaffold compound displayed excellent metabolic stability and was highly effective in suppressing solid tumor growth in vivo. Furthermore, the effectiveness of this compound ...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید