نتایج جستجو برای: endocannabinoid

تعداد نتایج: 3595  

2008
M. A. STORR B. YÜCE C. N. ANDREWS K. A. SHARKEY

Irritable bowel syndrome (IBS) is a spectrum of disorders characterized by abdominal discomfort and pain, associated with altered bowel habits. Though gut motility, secretion and sensation may be altered in patients with IBS, the pathophysiology of this condition remains to be fully understood. The endocannabinoid system is involved in the regulation of numerous gastrointestinal functions inclu...

Journal: :Chemistry & biology 2009
Kay Ahn Douglas S Johnson Mauro Mileni David Beidler Jonathan Z Long Michele K McKinney Eranthie Weerapana Nalini Sadagopan Marya Liimatta Sarah E Smith Scott Lazerwith Cory Stiff Satwik Kamtekar Keshab Bhattacharya Yanhua Zhang Stephen Swaney Keri Van Becelaere Raymond C Stevens Benjamin F Cravatt

Endocannabinoids are lipid signaling molecules that regulate a wide range of mammalian behaviors, including pain, inflammation, and cognitive/emotional state. The endocannabinoid anandamide is principally degraded by the integral membrane enzyme fatty acid amide hydrolase (FAAH), and there is currently much interest in developing FAAH inhibitors to augment endocannabinoid signaling in vivo. Her...

Journal: :Journal of neurobiology 2004
Benjamin F Cravatt Aron H Lichtman

The analgesic properties of exogenous cannabinoids have been recognized for many years and suggest a regulatory role for the endogenous cannabinoid ("endocannabinoid") system in mammalian nociceptive pathways. The endocannabinoid system includes: (1) at least two families of lipid signaling molecules, the N-acyl ethanolamines (e.g., anandamide) and the monoacylglycerols (e.g., 2-arachidonoyl gl...

Journal: :Molecular human reproduction 2013
Hyun-Ah Oh Sojung Kwon Soyoung Choi Hyejin Shin Kwang Ho Yoon Wan Jong Kim Hyunjung Jade Lim

Endocannabinoid signaling plays various roles in directing reproductive processes. Mouse embryos are shown to express high levels of CB1 receptor (CB1R). Low concentrations of anandamide stimulate embryo growth and implantation but at higher concentrations it adversely affects implantation. We tested the hypothesis that high levels of endocannabinoids cause autophagic activation and cell death ...

2014
Alán Alpár Giuseppe Tortoriello Daniela Calvigioni Micah J Niphakis Ivan Milenkovic Joanne Bakker Gary A Cameron János Hanics Claudia V Morris János Fuzik Gabor G Kovacs Benjamin F Cravatt John G Parnavelas William D Andrews Yasmin L Hurd Erik Keimpema Tibor Harkany

Local environmental cues are indispensable for axonal growth and guidance during brain circuit formation. Here, we combine genetic and pharmacological tools, as well as systems neuroanatomy in human fetuses and mouse models, to study the role of endocannabinoid and Slit/Robo signalling in axonal growth. We show that excess 2-arachidonoylglycerol, an endocannabinoid affecting directional axonal ...

Journal: :European journal of pharmacology 2014
Keith A Sharkey Nissar A Darmani Linda A Parker

Nausea and vomiting (emesis) are important elements in defensive or protective responses that animals use to avoid ingestion or digestion of potentially harmful substances. However, these neurally-mediated responses are at times manifested as symptoms of disease and they are frequently observed as side-effects of a variety of medications, notably those used to treat cancer. Cannabis has long be...

2008
Andreas Zimmer

Introduction Although the endocannabinoid system (ECS) is best known for its important neuromodulatory role, it has become apparent in recent years that the physiology of almost every organ is affected by the ECS. This is especially true under pathological conditions, in which an up-regulation of the expression of cannabinoid receptors and increased endocannabinoid production can often be obser...

Journal: :Journal of neurophysiology 2009
William M Connelly Matthew J Baggott

Endocannabinoids are lipid retrograde messengers that can be released by postsynaptic depolarization and/or activation of certain metabotropic receptors. We review a recent report that activation of metabotropic 5-HT2 receptors by endogenous serotonin induces the release of endocannabinoids in the olivary nucleus and suppresses glutamatergic input through a presynaptic action. This serotonin-en...

Journal: :Neuroscience 2003
M Egertová B F Cravatt M R Elphick

Fatty acid amide hydrolase (FAAH) catalyses hydrolysis of the endocannabinoid arachidonoylethanolamide ("anandamide") in vitro and regulates anandamide levels in the brain. In the cerebellar cortex, hippocampus and neocortex of the rat brain, FAAH is located in the somata and dendrites of neurons that are postsynaptic to axon fibers expressing the CB(1) cannabinoid receptor [Proc R Soc Lond B 2...

Journal: :The Journal of neuroscience : the official journal of the Society for Neuroscience 2005
David A Karanian Queenie B Brown Alexandros Makriyannis Therese A Kosten Ben A Bahr

The endocannabinoid system has been suggested to elicit signals that defend against several disease states including excitotoxic brain damage. Besides direct activation with CB1 receptor agonists, cannabinergic signaling can be modulated through inhibition of endocannabinoid transport and fatty acid amide hydrolase (FAAH), two mechanisms of endocannabinoid inactivation. To test whether the tran...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید