نتایج جستجو برای: benzopyran

تعداد نتایج: 614  

Journal: :Acta Crystallographica Section E Structure Reports Online 2005

Journal: :The Journal of pharmacology and experimental therapeutics 2002
Elisabetta Galbiati Paola Lorenza Caruso Gabriele Amari Elisabetta Armani Silvia Ghirardi Maurizio Delcanale Maurizio Civelli

We have discovered a new, nonsteroidal, estrogen agonist/antagonist, 3-phenyl-4-[[4-[2-(1-piperidinyl)ethoxy]phenyl] methyl]-2H-1-benzopyran-7-ol (CHF 4056). The aim of this study was to determine the effects of CHF 4056 on a series of parameters (body weight, uteri, serum cholesterol, and bones) that were previously shown to be sensitive to estrogens and to selective estrogen receptor modulato...

Journal: :Molecules 2015
Dmitry G Deryabin Anna A Tolmacheva

Quercus cortex (Oak bark) has been used in European folk medicine since medieval times for treatment of diarrhea, stomatitis, pharyngitis and skin inflammations. Its antimicrobial activity is a well-known therapeutic property of oak bark, and its novel anti-quorum sensing (QS) ability has also been described recently. In this study, we examined the bioactive compounds of Quercus cortex extract ...

Journal: :The Journal of neuroscience : the official journal of the Society for Neuroscience 2004
Kevin Park Jian-Min Luo Susan Hisheh Alan R Harvey Qi Cui

We have shown previously that intraocular elevation of cAMP using the cAMP analog 8-(4-chlorophenylthio)-cAMP (CPT-cAMP) failed to promote axonal regeneration of axotomized adult retinal ganglion cells (RGCs) into peripheral nerve (PN) grafts but significantly potentiated ciliary neurotrophic factor (CNTF)-induced axonal regeneration. Using the PN graft model, we now examine the mechanisms unde...

Journal: :The Journal of pharmacology and experimental therapeutics 2001
L Rënyi J L Evenden C J Fowler E Jerning D Kelder D Lake-Bakaar L G Larsson N Mohell M Sällemark S B Ross

The pharmacological properties of the 5-hydroxytryptamine (HT)(1A) receptor agonist (R)-3,4-dihydro-N-isopropyl-3-(N-isopropyl-N-propylamino)-2H-1-benzopyran-5-carboxamide (NAE-086) were examined with in vitro and in vivo techniques. Receptor binding studies demonstrated that NAE-086 was a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hip...

Journal: :BMC complementary medicine and therapies 2021

Abstract Background New agents for developing alternative or complementary medicine to treat the hepatitis C virus (HCV) are still needed due high rates of HCV infection globally and current limitations available treatments. Treatment with a combination direct acting antivirals have been shown be approximately 90% effective but will limited in future emergence drug resistance cost. The leaves M...

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