نتایج جستجو برای: ccr2b receptor inhibitors

تعداد نتایج: 746644  

Journal: :caspian journal of internal medicine 0
farshid oliaei shirin hushmand soraya khafri mahmoud baradaran

background: diabetic nephropathy is considered to be the most common cause of end stage renal disease (esrd). proteinuria is declared as the most marked risk factor in progression towards esrd. the aim of this study was to evaluate the efficacy of pentoxifylline for reduction of proteinuria in type ii diabetic patients. methods: from may 2007 to june 2008, this randomized clinical trial study w...

Journal: :ACS Medicinal Chemistry Letters 2016

Journal: :Proceedings for Annual Meeting of The Japanese Pharmacological Society 2018

Journal: :World Journal of Biological Chemistry 2017

Journal: :Archives of Pharmacy Practice 2021

Hypertension is considered a major health problem around the world. It’s associated with increasing risk of mortality due to its complication which has great impact on patient’s life quality. Angiotensin Receptor Blocker been widely used manage hypertension, especially if diabetes coexists and patient less tolerable angiotensin-converting enzyme inhibitors. In particular, telmisarta...

2017
Catriona E. Barker Sarah Thompson Graeme O’Boyle Hugues Lortat-Jacob Neil S. Sheerin Simi Ali John A. Kirby

Chemokines promote leukocyte recruitment during inflammation. The oxidative burst is an important effector mechanism, this leads to the generation of reactive nitrogen species (RNS), including peroxynitrite (ONOO). The current study was performed to determine the potential for nitration to alter the chemical and biological properties of the prototypical CC chemokine, CCL2. Immunofluorescence wa...

Journal: :Molecular cancer therapeutics 2011
Matthew Squires George Ward Gordan Saxty Valerio Berdini Anne Cleasby Peter King Patrick Angibaud Tim Perera Lynsey Fazal Douglas Ross Charlotte Griffiths Jones Andrew Madin Rajdeep K Benning Emma Vickerstaffe Alistair O'Brien Martyn Frederickson Michael Reader Christopher Hamlett Michael A Batey Sharna Rich Maria Carr Darcey Miller Ruth Feltell Abarna Thiru Susanne Bethell Lindsay A Devine Brent L Graham Andrew Pike Jose Cosme Edward J Lewis Eddy Freyne John Lyons Julie Irving Christopher Murray David R Newell Neil T Thompson

We describe here the identification and characterization of 2 novel inhibitors of the fibroblast growth factor receptor (FGFR) family of receptor tyrosine kinases. The compounds exhibit selective inhibition of FGFR over the closely related VEGFR2 receptor in cell lines and in vivo. The pharmacologic profile of these inhibitors was defined using a panel of human tumor cell lines characterized fo...

Journal: :Journal of the American College of Cardiology 1999
H P Brunner-La Rocca G Vaddadi M D Esler

One possible intervention to interrupt the deleterious effects of the renin-angiotensin system is suppression of angiotensin II (Ang II) formation by inhibition of angiotensin-converting enzyme (ACE). However, ACE inhibition incompletely suppresses Ang II formation and also leads to accumulation of bradykinin. Angiotensin II type 1 (AT1) receptors are believed to promote the known deleterious e...

2013
John Gerich

Postprandial plasma glucose concentrations are an important contributor to glycemic control. There is evidence suggesting that postprandial hyperglycemia may be an independent risk factor for cardiovascular disease. Glucagon-like peptide-1 (GLP-1) receptor agonists and dipeptidyl peptidase-4 (DPP-4) inhibitors are antidiabetic agents that predominantly reduce postprandial plasma glucose levels....

Journal: :The Journal of Experimental Medicine 1993
A Sarin D H Adams P A Henkart

The hypothesis that cytoplasmic proteases play a functional role in programmed cell death was tested by examining the effect of protease inhibitors on the T cell receptor-mediated death of the 2B4 murine T cell hybridoma and activated T cells. The cysteine protease inhibitors trans-epoxysuccininyl-L-leucylamido-(4-guanidino) butane (E-64) and leupeptin, the calpain selective inhibitor acetyl-le...

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