نتایج جستجو برای: conformationally restricted

تعداد نتایج: 119548  

Journal: :Angewandte Chemie 2004
Valentin Wittmann Sonja Seeberger

Natural and synthetic polyvalent ligands can act as inhibitors of biological processes or as effectors of signal-transduction pathways. 2] In the case of carbohydrate–lectin interactions, polyvalency is of particular importance because individual carbohydrate epitopes are usually bound with only weak affinity and often broad specificity. The potency of a polyvalent inhibitor depends on the spat...

Journal: :The Journal of biological chemistry 1988
G Lin J Noel W Loffredo H Z Stable M D Tsai

A great mystery in the mechanism of phospholipase A2 (PLA2) and many other lipolytic enzymes is the "interfacial activation" induced by micellar but not monomeric substrates. Equally mysterious is the lack of interfacial activation in bee venom PLA2, as opposed to PLA2s from pancreas and other sources. We have probed these problems using the conformationally restricted short-chain cyclopentano-...

2011
Raju Sunagar Vidiya Ramachandran Melina Georgousakis Kadaba S. Sriprakash Melkote S. Shaila

A peptide (J14) containing conformationally restricted epitopes from the M protein of group A streptococcus (GAS) is capable of eliciting protective immune response against GAS infection. However, the protective response may be lost possibly due to its weak secondary-structure when the antigen is fused with other antigens in a recombinant polyepitope vaccine construct. We previously showed that...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 2017
Yongfei Cai Selen Karaca-Griffin Jia Chen Sai Tian Nicholas Fredette Christine E Linton Sophia Rits-Volloch Jianming Lu Kshitij Wagh James Theiler Bette Korber Michael S Seaman Stephen C Harrison Andrea Carfi Bing Chen

The extraordinary genetic diversity of the HIV-1 envelope spike [Env; trimeric (gp160)3, cleaved to (gp120/gp41)3] poses challenges for vaccine development. Envs of different clinical isolates exhibit different sensitivities to antibody-mediated neutralization. Envs of difficult-to-neutralize viruses are thought to be more stable and conformationally homogeneous trimers than those of easy-to-ne...

2007
Melissa Maderia Shilpa Shenoy Que N. Van Victor E. Marquez Joseph J. Barchi

The biophysical properties of oligodeoxyribonucleotides (ODNs) selectively modified with conformationally 'locked' bicyclo[3.1.0]hexane pseudosugars (Maier,M.A., Choi,Y., Gaus,H., Barchi,J.J. Jr, Marquez,V.E., Manoharan,M. (2004) Synthesis and characterization of oligonucleotides containing conformationally constrained bicyclo[3.1.0]hexane pseudosugar analogs Nucleic Acids Res., 32, 3642-3650) ...

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