نتایج جستجو برای: pik3ca

تعداد نتایج: 2433  

Journal: :British journal of haematology 2014
Claudia Hofmann Thorsten Stühmer Nadine Schmiedl Reinhard Wetzker Anja Mottok Andreas Rosenwald Christian Langer Josip Zovko Manik Chatterjee Hermann Einsele Ralf C Bargou Torsten Steinbrunn

Constitutive phosphatidylinositide 3-kinase (PI3K) signalling has been implicated in multiple myeloma (MM) pathophysiology and is regarded as an actionable target for pharmacological intervention. Isoform-specific PI3K inhibition may offer the most focused treatment approach and could result in greater clinical efficacy and reduced side effects. We therefore performed isoform-specific knockdown...

2013
Heesue Kim Cheol-Keun Park Su Jin Lee Sun Young Rha Kyu Hyun Park Ho Yeong Lim

PURPOSE Phosphatidylinositol 3-kinases/AKT pathway plays a pivotal role in hepatocellular carcinoma (HCC). Mutant PIK3CA, encoding the p110a catalytic subunit, stimulates the AKT pathway and promotes cell growth in various cancers. PIK3CA mutation rate has been usually reported as low frequency (<5%) in HCC except one report from Korea with 35.6%. Therefore, we investigated the frequency of PIK...

Journal: :Cancer research 2008
Katsutoshi Oda Jennifer Okada Luika Timmerman Pablo Rodriguez-Viciana David Stokoe Keiko Shoji Yuji Taketani Hiroyuki Kuramoto Zachary A Knight Kevan M Shokat Frank McCormick

Mutations in genes functioning in different pathways frequently occur together in the same cancer, whereas mutations in the same pathway tend to be mutually exclusive. However, the majority of colon, breast, and endometrial cancers that possess mutations in PIK3CA, the catalytic subunit p110alpha of phosphatidylinositol 3'-kinase (PI3K), also possess mutations or alterations in genes upstream o...

Journal: :Cancer research 2013
Grace M Wang Hong Yuen Wong Hiroyuki Konishi Brian G Blair Abde M Abukhdeir John P Gustin D Marc Rosen Samuel Ray Denmeade Zeshaan Rasheed William Matsui Joseph P Garay Morassa Mohseni Michaela J Higgins Justin Cidado Danijela Jelovac Sarah Croessmann Rory L Cochran Sivasundaram Karnan Yuko Konishi Akinobu Ota Yoshitaka Hosokawa Pedram Argani Josh Lauring Ben Ho Park

The selective pressures leading to cancers with mutations in both KRAS and PIK3CA are unclear. Here, we show that somatic cell knockin of both KRAS G12V and oncogenic PIK3CA mutations in human breast epithelial cells results in cooperative activation of the phosphoinositide 3-kinase (PI3K) and mitogen-activated protein kinase (MAPK) pathways in vitro, and leads to tumor formation in immunocompr...

2014
Andrea Casadei Gardini Laura Capelli Paola Ulivi Massimo Giannini Eva Freier Stefano Tamberi Emanuela Scarpi Alassandro Passardi Wainer Zoli Angela Ragazzini Dino Amadori Giovanni Luca Frassineti

Anti-EGFR therapy appears to be a potential treatment option for squamous cell anal carcinoma (SCAC). KRAS mutation is a rare event in SCAC, indicating the absence of the principal mechanism of resistance to this type of therapy. However, no information is available from the literature regarding the status of BRAF or PIK3CA in this cancer type. We analysed KRAS, BRAF and PIK3CA status in SCAC p...

Journal: :Anticancer research 2009
Xiuju Sun Jian Huang Taku Homma Daisuke Kita Helmut Klocker Georg Schafer Peter Boyle Hiroko Ohgaki

Alterations in the PIK3CA and PTEN genes were assessed in 40 prostate tumors (radical prostatectomy samples). Genetic analyses in glands of the highest Gleason pattern within each tumor revealed PIK3CA amplification in 13%, PIK3CA mutations in 3%, PTEN homozygous deletion in 13% and PTEN hemizygous deletion in 8% of the cases analyzed. Supporting the view that PTEN and PIK3CA act in the same PI...

Journal: :Cancer research 2014
Yi-Zhou Jiang Ke-Da Yu Jing Bao Wen-Ting Peng Zhi-Ming Shao

We investigated the loss of somatic mutations in TP53 and PIK3CA in breast cancer tissue after neoadjuvant chemotherapy (NCT) and the clinical relevance of the observed mutation profiles. Samples were derived from three cohorts: Cohort 1 consisting of 206 patients undergoing NCT with matched pre- and postchemotherapy tumor tissues; Cohort 2 consisting of 158 additional patients undergoing NCT; ...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2014
Julia A Beaver Danijela Jelovac Sasidharan Balukrishna Rory Cochran Sarah Croessmann Daniel J Zabransky Hong Yuen Wong Patricia Valda Toro Justin Cidado Brian G Blair David Chu Timothy Burns Michaela J Higgins Vered Stearns Lisa Jacobs Mehran Habibi Julie Lange Paula J Hurley Josh Lauring Dustin VanDenBerg Jill Kessler Stacie Jeter Michael L Samuels Dianna Maar Leslie Cope Ashley Cimino-Mathews Pedram Argani Antonio C Wolff Ben H Park

PURPOSE Detecting circulating plasma tumor DNA (ptDNA) in patients with early-stage cancer has the potential to change how oncologists recommend systemic therapies for solid tumors after surgery. Droplet digital polymerase chain reaction (ddPCR) is a novel sensitive and specific platform for mutation detection. EXPERIMENTAL DESIGN In this prospective study, primary breast tumors and matched p...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 2009
H B Salvesen S L Carter M Mannelqvist A Dutt G Getz I M Stefansson M B Raeder M L Sos I B Engelsen J Trovik E Wik H Greulich T H Bø I Jonassen R K Thomas T Zander L A Garraway A M Oyan W R Sellers K H Kalland M Meyerson L A Akslen R Beroukhim

Although 75% of endometrial cancers are treated at an early stage, 15% to 20% of these recur. We performed an integrated analysis of genome-wide expression and copy-number data for primary endometrial carcinomas with extensive clinical and histopathological data to detect features predictive of recurrent disease. Unsupervised analysis of the expression data distinguished 2 major clusters with s...

Journal: :Cancer research 2005
Milo Frattini Stefano Signoroni Silvana Pilotti Lucio Bertario Silvia Benvenuti Carlo Zanon Alberto Bardelli Marco A Pierotti

Phosphatidylinositol-3 phosphate kinase (PI3K) and phosphatase protein homologue to tensin (PTEN) are involved in cell signaling by catalyzing opposite reactions in the balance of phosphatidylinositol-3,4,5,-trisphosphate and are deregulated in many tumors. Recently, Saal et al. (1) reported that these two proteins are altered in a consistent fraction of breast cancers and, more importantly, th...

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