نتایج جستجو برای: natural compound

تعداد نتایج: 601460  

2013
Alessandra Mascarello Mattia Mori Louise Domeneghini Chiaradia-Delatorre Angela Camila Orbem Menegatti Franco Delle Monache Franco Ferrari Rosendo Augusto Yunes Ricardo José Nunes Hernán Terenzi Bruno Botta Maurizio Botta

Protein tyrosine phosphatase B (PtpB) is one of the virulence factors secreted into the host cell by Mycobacterium tuberculosis. PtpB attenuates host immune defenses by interfering with signal transduction pathways in macrophages and, therefore, it is considered a promising target for the development of novel anti-tuberculosis drugs. Here we report the discovery of natural compound inhibitors o...

Journal: :Molecules 2017
Murali Annamalai Stanimira Hristeva Martyna Bielska Raquel Ortega Kamal Kumar

Despite the great contribution of natural products in the history of successful drug discovery, there are significant limitations that persuade the pharmaceutical industry to evade natural products in drug discovery research. The extreme scarcity as well as structural complexity of natural products renders their practical synthetic access and further modifications extremely challenging. Althoug...

2017
Qian Lin Leina Ma Zhantao Liu Zhihong Yang Jin Wang Jia Liu Guohui Jiang

Unlike genetics, epigenetics involves the modification of genome without changes in DNA sequences, including DNA methylation, histone modification, chromatin remodeling and noncoding RNA regulation. MicroRNA (miRNA), a member of noncoding RNAs superfamily, participates in RNA interference through a unique mechanism. Currently, microRNAs have been found to be regulated by some natural compounds....

Journal: :Journal of applied biology and biotechnology 2021

Astaxanthin: An algae-based natural compound with a potential role in human health-promoting effect: updated comprehensive reviewJinu Medhi, Mohan Chandra Kalita

Journal: :Chemical communications 2015
Zhangfeng Zhong Li-Juan Liu Zhi-Qiang Dong Lihua Lu Modi Wang Chung-Hang Leung Dik-Lung Ma Yitao Wang

We report herein the identification of an immunomodulatory natural product-like compound as a direct inhibitor of TLR1-TLR2 heterodimerization. Compound suppressed TNF-α and IL-6 secretion in Pam3CSK4-induced macrophages. Moreover, compound inhibited the phagocytic activity of macrophages, presumably through modulation of TLR1-TLR2 signaling and inactivation of NF-κB. Molecular docking revealed...

Journal: :American Journal of Physiology-Lung Cellular and Molecular Physiology 2010

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