نتایج جستجو برای: chemotypes

تعداد نتایج: 676  

2008
Tridib Mahapatra Tapas Das Samik Nanda

Article history: Received 2 October 2008 Accepted 22 October 2008 0957-4166/$ see front matter 2008 Elsevier Ltd. A doi:10.1016/j.tetasy.2008.10.024 * Corresponding author. E-mail address: [email protected] (S. N Novel multifunctional chemotypes based on a-tetralone, a-indanone, and chromanone have been synthesized by a chemo-enzymatic approach by applying an enzymatic irreversible tr...

Journal: :Current opinion in structural biology 2004
Jeanne A Hardy James A Wells

The discovery of new allosteric sites generates opportunities for the identification of novel pharmaceuticals and increases our understanding of basic biological processes. Increasingly, allosteric sites are being discovered in various families of proteins by several methods, paving the way for the development of entirely new classes of drugs with a wide range of chemotypes. New allosteric site...

2015
Anna Barnard Kérya Long Heather L. Martin Jennifer A. Miles Thomas A. Edwards Darren C. Tomlinson Andrew Macdonald Andrew J. Wilson

Inhibition of protein-protein interactions (PPIs) represents a major challenge in chemical biology and drug discovery. α-Helix mediated PPIs may be amenable to modulation using generic chemotypes, termed "proteomimetics", which can be assembled in a modular manner to reproduce the vectoral presentation of key side chains found on a helical motif from one partner within the PPI. In this work, it...

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