S derivatives of γ-aminobutyric acid (GABA), the principal inhibitory neurotransmitter in the mammalian brain, have been extensively used for the treatment of several nervous system disorders including epilepsy, neuropathic pain, anxiety, and social phobia. Several drugs such as Gabapentin and Pregabalin have achieved rapid success in the past two decades. The use of an enzymatic kinetic resolu...
