نتایج جستجو برای: hiv fusion inhibitors

تعداد نتایج: 504964  

Journal: :Journal of virology 2005
Surender Khurana Michael Kennedy Lisa R King Hana Golding

CCR5 is the major coreceptor for human immunodeficiency virus (HIV) infection. The murine monoclonal antibody (MAb) 2D7, which recognizes a conformation-dependent epitope in the second extracellular loop of CCR5, is one of the most potent inhibitors of R5 virus cell entry. However, attempts to humanize 2D7 for in vivo human use have been unsuccessful so far. A filamentous phage library expressi...

2014
Andrea C Tricco Jesmin Antony Veroniki A Angeliki Huda Ashoor Brian Hutton Brenda R Hemmelgarn David Moher Yaron Finkelstein Kevin Gough Sharon E Straus

BACKGROUND Antiretroviral therapy reduces mother-to-child transmission of human immunodeficiency virus (HIV) during pregnancy, delivery, and breastfeeding. However, these agents have been associated with preterm birth, anemia and low birth weight. We aim to evaluate the comparative safety and effectiveness of the use of antiretroviral drugs among HIV-infected women and the effects on their infa...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 1998
M Pritsker P Jones R Blumenthal Y Shai

Recent studies demonstrated that a synthetic fusion peptide of HIV-1 self-associates in phospholipid membranes and inhibits HIV-1 envelope glycoprotein-mediated cell fusion, presumably by interacting with the N-terminal domain of gp41 and forming inactive heteroaggregates [Kliger, Y., Aharoni, A., Rapaport, D., Jones, P., Blumenthal, R. & Shai, Y. (1997) J. Biol. Chem. 272, 13496-13505]. Here, ...

Journal: :Bioorganic & Medicinal Chemistry 2021

Non-nucleoside reverse transcriptase inhibitors (NNRTIs) are widely used in combination therapies against HIV-1. However, emergent and transmitted drug resistance compromise their efficacy the clinical setting. Y181C is selected patients receiving nevirapine, etravirine rilpivirine, together with K103N most prevalent NNRTI-associated mutation HIV-infected patients. Herein, we report on design, ...

Journal: :Current Biology 1997
M Loetscher A Amara E Oberlin N Brass D. F Legler P Loetscher M D’Apuzzo E Meese D Rousset J-L Virelizier M Baggiolini F Arenzana-Seisdedos B Moser

BACKGROUND Chemokines bind to specific receptors and mediate leukocyte migration to sites of inflammation. Recently, some chemokine receptors, notably CXCR4 and CCR5, have been shown to be essential fusion factors on target cells for infection by human immunodeficiency virus (HIV); the chemokines bound by these receptors have also been shown to act as potent inhibitors of HIV infection. Here, w...

Journal: :International Journal of Antimicrobial Agents 2021

• Despite successful antiretroviral therapy, patients with human immunodeficiency virus (HIV) could develop multi-class drug resistance (MDR) Data about the prevalence of HIV-MDR are scanty and results unclear A significant decline in over between 1998 2018 was observed Nowadays, still occurs, although at a lower rate Management infected by MDR viruses is critical issue HIV therapy (ART), can (...

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