نتایج جستجو برای: nitroreductase

تعداد نتایج: 396  

Journal: :Molecules 2009
Gabi U Dachs Michelle A Hunt Sophie Syddall Dean C Singleton Adam V Patterson

Gene directed enzyme prodrug therapy (GDEPT) of cancer aims to improve the selectivity of chemotherapy by gene transfer, thus enabling target cells to convert nontoxic prodrugs to cytotoxic drugs. A zone of cell kill around gene-modified cells due to transfer of toxic metabolites, known as the bystander effect, leads to tumour regression. Here we discuss the implications of either striving for ...

Journal: :Fungal genetics and biology : FG & B 2011
Tünde Pusztahelyi Eva Klement Emilia Szajli József Klem Márton Miskei Zsolt Karányi Tamás Emri Szilvia Kovács Gyula Orosz Kornél L Kovács Katalin F Medzihradszky Rolf A Prade István Pócsi

Under long-term oxidative stress caused by menadione sodium bisulfite, genome-wide transcriptional and proteome-wide translational changes were compared in Aspergillus nidulans vegetative cells. The comparison of proteomic and DNA microarray expression data demonstrated that global gene expression changes recorded with either flip-flop or dendrimer cDNA labeling techniques supported proteome ch...

2016
Stephen Patterson Susan Wyllie Suzanne Norval Laste Stojanovski Frederick Rc Simeons Jennifer L Auer Maria Osuna-Cabello Kevin D Read Alan H Fairlamb

There is an urgent requirement for safe, oral and cost-effective drugs for the treatment of visceral leishmaniasis (VL). We report that delamanid (OPC-67683), an approved drug for multi-drug resistant tuberculosis, is a potent inhibitor of Leishmania donovani both in vitro and in vivo. Twice-daily oral dosing of delamanid at 30 mg kg(-1) for 5 days resulted in sterile cures in a mouse model of ...

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