نتایج جستجو برای: phthalazine

تعداد نتایج: 192  

Journal: :The American journal of physiology 1953
I H PAGE J W McCUBBIN

ER~TONIN S (s-hydroxytryptamine) has only Bouckaert and Moraes (8) to reverse the vasorecently been isolated, synthesized and constrictor activity of defibrinated blood in available in quantities sufficient to study perfusion experiments; its action against pure its pharmacologic actions. In a brief span of serotonin is evaluated here; e) Pitressin tends time several publications have appeared ...

Journal: :iranian journal of catalysis 2015
mahdieh chegeni ardeshier khazaei sadegh rahmati mohammad hossein fekri

in this report, synthesis, characterization and application of silica perchloric acid nanosphere as a novel and heterogeneous catalyst is described. these nanospheres have been characterized by xrd, ft-ir, bet and tga spectra and also by sem and tem images. the results show that it has a spherical shape and the particles size are between 75 and 100 nm. the catalytic activity has been investigat...

Sulfonated magnetic nanoparticles (SO3H-Fe3O4@SiO2 MNPs) have been explored as an efficient, cost-effective, and recyclable nanocatalyst for the facile synthesis of 3,4-dihydro-2H-indazolo[1,2-b]phthalazin-1,6,11(13H)-triones through a one-pot three-component reaction between aldehydes, dimedone, and phthalhydrazide under mild and green (solvent-f...

2009
John R. Atack Karen A. Maubach Keith A. Wafford Desmond O’Connor A. David Rodrigues David C. Evans F. David Tattersall Mark S. Chambers Angus M. MacLeod Wai-Si Eng Christine Ryan Eric Hostetler Sandra M. Sanabria Raymond E. Gibson Stephen Krause H. Donald Burns Richard J. Hargreaves Nancy G. B. Agrawal Ruth M. McKernan M. Gail Murphy Kevin Gingrich Gerard R. Dawson Donald G. Musson Kevin J. Petty

3-tert-Butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4triazol-5-ylmethoxy)-pyrazolo[1,5-d][1,2,4]triazine (MRK-016) is a pyrazolotriazine with an affinity of between 0.8 and 1.5 nM for the benzodiazepine binding site of native rat brain and recombinant human 1-, 2-, 3-, and 5-containing GABAA receptors. It has inverse agonist efficacy selective for the 5 subtype, and this 5 inverse agonism...

2008

Aldehyde oxidase-mediated oxidation of N-methylnicotinamide to N-methyl-2-pyridine-5-carboxamide (2-PY) and N-methyl-4pyridone-5-carboxamide (4-PY) in chimeric mice constructed by transplanting human hepatocytes into urokinase-type plasminogen activator-transgenic severe combined immunodeficient mice was examined in vivo and in vitro. The activity in liver cytosol of chimeric mice with a high r...

2008

Aldehyde oxidase-mediated oxidation of N-methylnicotinamide to N-methyl-2-pyridine-5-carboxamide (2-PY) and N-methyl-4pyridone-5-carboxamide (4-PY) in chimeric mice constructed by transplanting human hepatocytes into urokinase-type plasminogen activator-transgenic severe combined immunodeficient mice was examined in vivo and in vitro. The activity in liver cytosol of chimeric mice with a high r...

2008

Aldehyde oxidase-mediated oxidation of N-methylnicotinamide to N-methyl-2-pyridine-5-carboxamide (2-PY) and N-methyl-4pyridone-5-carboxamide (4-PY) in chimeric mice constructed by transplanting human hepatocytes into urokinase-type plasminogen activator-transgenic severe combined immunodeficient mice was examined in vivo and in vitro. The activity in liver cytosol of chimeric mice with a high r...

2008

Aldehyde oxidase-mediated oxidation of N-methylnicotinamide to N-methyl-2-pyridine-5-carboxamide (2-PY) and N-methyl-4pyridone-5-carboxamide (4-PY) in chimeric mice constructed by transplanting human hepatocytes into urokinase-type plasminogen activator-transgenic severe combined immunodeficient mice was examined in vivo and in vitro. The activity in liver cytosol of chimeric mice with a high r...

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