نتایج جستجو برای: antiparasitic drugs

تعداد نتایج: 225369  

Journal: :The Journal of biological chemistry 2009
Iain D Kerr Ji H Lee Christopher J Farady Rachael Marion Mathias Rickert Mohammed Sajid Kailash C Pandey Conor R Caffrey Jennifer Legac Elizabeth Hansell James H McKerrow Charles S Craik Philip J Rosenthal Linda S Brinen

Cysteine proteases of the papain superfamily are implicated in a number of cellular processes and are important virulence factors in the pathogenesis of parasitic disease. These enzymes have therefore emerged as promising targets for antiparasitic drugs. We report the crystal structures of three major parasite cysteine proteases, cruzain, falcipain-3, and the first reported structure of rhodesa...

2000
OLIVER KAYSER ALBRECHT F. KIDERLEN SIMON L. CROFT

Pharmaceutical research in natural products represents a major strategy for discovering and developing new drugs. The use of medicinal plants for the treatment of parasitic diseases is well known and documented since ancient times e.g. by the use of Cinchona succiruba (Rubiaceae) as an antimalarial. This chapter provides a comprehensive review of the latest results in the field of antiparasitic...

Journal: :Antimicrobial agents and chemotherapy 2006
Jacqueline A Upcroft Linda A Dunn Janelle M Wright Kamel Benakli Peter Upcroft Patrice Vanelle

Metronidazole (Mz)-resistant Giardia and Trichomonas were inhibited by 1 of 30 new 5-nitroimidazole drugs. Another five drugs were effective against some but not all of the Mz-resistant parasites. This study provides the incentive for the continued design of 5-nitroimidazole drugs to bypass cross-resistance among established 5-nitromidazole antiparasitic drugs.

Journal: :Molecules 2013
Ifedayo Victor Ogungbe William N Setzer

Neglected Tropical Diseases (NTDs), like leishmaniasis, are major causes of mortality in resource-limited countries. The mortality associated with these diseases is largely due to fragile healthcare systems, lack of access to medicines, and resistance by the parasites to the few available drugs. Many antiparasitic plant-derived isoprenoids have been reported, and many of them have good in vitro...

2013
Dieudonné Ndjonka Ludmila Nakamura Rapado Ariel M. Silber Eva Liebau Carsten Wrenger

Infectious diseases caused by parasites are a major threat for the entire mankind, especially in the tropics. More than 1 billion people world-wide are directly exposed to tropical parasites such as the causative agents of trypanosomiasis, leishmaniasis, schistosomiasis, lymphatic filariasis and onchocerciasis, which represent a major health problem, particularly in impecunious areas. Unlike mo...

Journal: :Brazilian journal of biology = Revista brasleira de biologia 2016
G F Ferreira T M Freitas C L Gonçalves J F Mendes J N Vieira J P Villareal P S Nascente

The use of biological agents has been intensified in recent years against eggs and larvae of gastrointestinal nematodes as an alternative control method in pasture plant health management, with the concomitant use with antiparasitic drugs still occurring. The aim of this study was to test the in vitro activity of the following antiparasitic drugs: Ivermectin and albendazole against the followin...

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