نتایج جستجو برای: gdc

تعداد نتایج: 840  

Journal: :AJNR. American journal of neuroradiology 1998
D F Kallmes M H Kallmes H J Cloft J E Dion

PURPOSE We calculated the incremental cost-utility ratio for Guglielmi detachable coil (GDC) embolization versus no therapy for unruptured intracranial aneurysms considered inappropriate for surgical clipping procedures. METHODS Decision tree and Markov analyses that employ cohort simulation were applied to determine the incremental cost-utility ratio of GDC embolization versus no therapy for...

Journal: :AJNR. American journal of neuroradiology 2012
L Pierot C Cognard F Ricolfi R Anxionnat

BACKGROUND AND PURPOSE Matrix coils have been developed to prevent aneurysm recanalization. Midterm anatomic results in a prospective multicenter consecutive series including patients treated with GDC or Matrix coils for ruptured aneurysms are presented. MATERIALS AND METHODS Five hundred seventeen patients harboring ruptured aneurysms were treated with GDC (276 patients) or Matrix coils (241...

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2016
Laurent Salphati Bruno Alicke Timothy P Heffron Sheerin Shahidi-Latham Merry Nishimura Tim Cao Richard A Carano Jonathan Cheong Joan Greve Hartmut Koeppen Shari Lau Leslie B Lee Michelle Nannini-Pepe Jodie Pang Emile G Plise Cristine Quiason Linda Rangell Xiaolin Zhang Stephen E Gould Heidi S Phillips Alan G Olivero

Glioblastoma multiforme (GBM) is the most common primary brain tumor in adults. Limited treatment options have only marginally impacted patient survival over the past decades. The phophatidylinositol 3-kinase (PI3K) pathway, frequently altered in GBM, represents a potential target for the treatment of this glioma. 5-(6,6-Dimethyl-4-morpholino-8,9-dihydro-6H-[1,4]oxazino[4,3-e]purin-2-yl)pyrimid...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2011
Richard A Graham Bert L Lum Sravanthi Cheeti Jin Yan Jin Karin Jorga Daniel D Von Hoff Charles M Rudin Josina C Reddy Jennifer A Low Patricia M Lorusso

PURPOSE In a phase I trial for patients with refractory solid tumors, hedgehog pathway inhibitor vismodegib (GDC-0449) showed little decline in plasma concentrations over 7 days after a single oral dose and nonlinearity with respect to dose and time after single and multiple dosing. We studied the role of GDC-0449 binding to plasma protein alpha-1-acid glycoprotein (AAG) to better understand th...

2013
Jie Lin Deepak Sampath Michelle A. Nannini Brian B. Lee Michael Degtyarev Jason Oeh Heidi Savage Zhengyu Guan Rebecca Hong Robert Kassees Leslie B. Lee Tyler Risom Stefan Gross Bianca M. Liederer Hartmut Koeppen Nicholas J. Skelton Jeffrey J. Wallin Marcia Belvin Elizabeth Punnoose Lori S. Friedman Kui Lin

Purpose:We describe the preclinical pharmacology and antitumor activity of GDC-0068, a novel highly selective ATP-competitive pan-Akt inhibitor currently in clinical trials for the treatment of human cancers. Experimental Design: The effect of GDC-0068 on Akt signaling was characterized using specific biomarkers of the Akt pathway, and response to GDC-0068 was evaluated in human cancer cell lin...

2015
Jasleen K. Sodhi Susan Wong Donald S. Kirkpatrick Lichuan Liu S. Cyrus Khojasteh Cornelis E. C. A. Hop John T. Barr Jeffrey P. Jones Jason S. Halladay

GDC-0834, a Bruton’s tyrosine kinase inhibitor investigated as a potential treatment of rheumatoid arthritis, was previously reported to be extensively metabolized by amide hydrolysis such that no measurable levels of this compound were detected in human circulation after oral administration. In vitro studies in human liver cytosol determined that GDC-0834 (R)-N-(3-(6-(4-(1,4-dimethyl-3-oxopipe...

This current study reports preparation of Nickel-Gadolinium doped Ceria (Ni-GDC) composite via controlled unidirectional freeze casting of aqueous-based GDC slurry completed with nickel infiltrated into the porous GDC samples. Gadolinium doped ceria powder prepared by gel-combustion synthesis method. The oxide powder was confirmed to be the fluorite-structured of Ce0.8Gd0.2O1.9 solid solution b...

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Gadanium doped cerium oxide ceramic (GDC) is widely used as solid electrolytes in solid oxide fuel cells because of its high oxygen ion conductivity. In this study, the effect of addition of nano CuO as a sintering aid on the properties of GDC electrolyte were investigated. For this purpose, 0.2, 0.5, and 1% mole of nano Cuo was added to GDC ceramics, which was synthesized by the solid-state me...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2016
Zachary S Zumsteg Natasha Morse Gabriel Krigsfeld Gaorav Gupta Daniel S Higginson Nancy Y Lee Luc Morris Ian Ganly Stephan L Shiao Simon N Powell Christine H Chung Maurizio Scaltriti José Baselga

PURPOSE ActivatingPIK3CAgenomic alterations are frequent in head and neck squamous cell carcinoma (HNSCC), and there is an association between phosphoinositide 3-kinase (PI3K) signaling and radioresistance. Hence, we investigated the therapeutic efficacy of inhibiting PI3K with GDC-0032, a PI3K inhibitor with potent activity against p110α, in combination with radiation in HNSCC. EXPERIMENTAL ...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2013
Giuseppe Floris Agnieszka Wozniak Raf Sciot Haifu Li Lori Friedman Thomas Van Looy Jasmien Wellens Peter Vermaelen Christophe M Deroose Jonathan A Fletcher Maria Debiec-Rychter Patrick Schöffski

PURPOSE Oncogenic signaling in gastrointestinal stromal tumors (GIST) is sustained via PI3K/AKT pathway. We used a panel of six GIST xenograft models to assess efficacy of GDC-0941 as single agent or in combination with imatinib (IMA). EXPERIMENTAL DESIGN Nude mice (n = 136) were grafted bilaterally with human GIST carrying diverse KIT mutations. Mice were orally dosed over four weeks, groupe...

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