نتایج جستجو برای: salicylanilides

تعداد نتایج: 35  

2016
Major Gooyit Kim D. Janda

Prolonged use of broad-spectrum antibiotics disrupts the indigenous gut microbiota, which consequently enables toxigenic Clostridium difficile species to proliferate and cause infection. The burden of C. difficile infections was exacerbated with the outbreak of hypervirulent strains that produce copious amounts of enterotoxins and spores. In recent past, membrane-active agents have generated a ...

Journal: :Molecules 2012
Martin Krátký Jarmila Vinšová Jiřina Stolaříková

The increasing emergence especially of drug-resistant tuberculosis has led to a strong demand for new anti-tuberculosis drugs. Eighteen salicylanilide benzoates were evaluated for their inhibition potential against Mycobacterium tuberculosis, Mycobacterium avium and two strains of Mycobacterium kansasii; minimum inhibitory concentration values ranged from 0.5 to 16 μmol/L. The most active...

Journal: :Molecules 2010
Jan Otevrel Zuzana Mandelova Matus Pesko Jiahui Guo Katarina Kralova Frantisek Sersen Marcela Vejsova Danuta S Kalinowski Zaklina Kovacevic Aidan Coffey Jozef Csollei Des R Richardson Josef Jampilek

In this study, a series of twelve ring-substituted salicylanilides and carbamoylphenylcarbamates were prepared and characterized. The compounds were analyzed using RP-HPLC to determine lipophilicity. They were tested for their activity related to the inhibition of photosynthetic electron transport (PET) in spinach (Spinacia oleracea L.) chloroplasts. Moreover, their site of action in the photos...

Journal: :Molecules 2012
Martin Krátký Jarmila Vinšová Nabila Guisado Rodriguez Jiřina Stolaříková

A series of eighteen novel esters of salicylanilides with benzenesulfonic acid were designed, synthesized and characterized by IR, ¹H-NMR and ¹³C-NMR. They were evaluated in vitro as potential antimycobacterial agents towards Mycobacterium tuberculosis, Mycobacterium avium and two strains of Mycobacterium kansasii. In general, the minimum inhibitory concentrations range from 1 to 500 µmol/L. Th...

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