نتایج جستجو برای: thiacetazone

تعداد نتایج: 60  

2013
Kamaleddin Haj Mohammad Ebrahim Tehrani Farzad Kobarfard Parisa Azerang Maryam Mehravar Zohreh Soleimani Ghazaleh Ghavami Soroush Sardari

In this work, we reported the synthesis and evaluation of antimycobacterial and antifungal activity of a series of thiocarbohydrazone derivatives which are thiacetazone congeners. The target compounds were synthesized in superior yields by reacting thiocarbohydrazide with different aromatic aldehydes and methyl ketones. Compounds 8, 19 and 25 were found to be the most potent derivatives, exhibi...

Journal: :Journal of Nepal Medical Association 1970

Journal: :Antimicrobial agents and chemotherapy 2003
Lanfranco Fattorini Dejiang Tan Elisabetta Iona Maurizio Mattei Federico Giannoni Lara Brunori Simona Recchia Graziella Orefici

The activity of moxifloxacin was enhanced by the addition of ethionamide but not by that of cycloserine, thiacetazone, capreomycin, para-aminosalicylic acid, or linezolid in BALB/c mice infected with a strain of Mycobacterium tuberculosis resistant to isoniazid, rifampin, and six other drugs. These observations are important for the therapy of multidrug-resistant tuberculosis.

Journal: :Bulletin of Pharmaceutical Sciences. Assiut 1988

Journal: :Tuberculosis and Respiratory Diseases 1968

In this work, we reported the synthesis and evaluation of antimycobacterial and antifungalactivity of a series of thiocarbohydrazone derivatives which are thiacetazone congeners. Thetarget compounds were synthesized in superior yields by reacting thiocarbohydrazide withdifferent aromatic aldehydes and methyl ketones. Compounds 8, 19 and 25 were found to bethe most potent derivatives, exhibiting...

Journal: :iranian journal of pharmaceutical research 0
kamaleddin haj mohammad ebrahim tehrani department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran. farzad kobarfard 1- department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran. 2- phytochemistry research center, shahid beheshti university of medical sciences, tehran, iran. parisa azerang drug design and bioinformatics unit, medical biotechnology department, biotechnology research center, tehran, pasteur institute, 13164, iran. maryam mehravar drug design and bioinformatics unit, medical biotechnology department, biotechnology research center, tehran, pasteur institute, 13164, iran. zohreh soleimani department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran. ghazaleh ghavami drug design and bioinformatics unit, medical biotechnology department, biotechnology research center, tehran, pasteur institute, 13164

in this work, we reported the synthesis and evaluation of antimycobacterial and antifungalactivity of a series of thiocarbohydrazone derivatives which are thiacetazone congeners. thetarget compounds were synthesized in superior yields by reacting thiocarbohydrazide withdifferent aromatic aldehydes and methyl ketones. compounds 8, 19 and 25 were found to bethe most potent derivatives, exhibiting...

Journal: :iranian journal of pharmaceutical research 0
marjan esfahani zade department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran. koroush omidi central research laboratories, shahid beheshti university of medical sciences, tehran, iran. joel kauffman department of chemistry and biochemistry, university of the sciences in philadelphia, philadelphia, pa, usa. shahram shahraki zahedani department of microbiology, school of medicine, zahedan university of medical sciences, zahedan, iran ali gudarzi department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran. salimeh amidi department of medicinal chemistry, school of pharmacy, shahid beheshti university of medical sciences, tehran, iran.

treatment of tuberculosis (tb) and the discovery of effective new anti tubercular drugs is one of the most urgent priorities in health organizations all around the world. in the present study, fluorinated analogs of some of the most important anti-tb agents such as p-aminosalicylic acid (pas), thiacetazone and pyrazinamide were synthesized and tested against tb. the fluorinated analog of thiace...

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