نتایج جستجو برای: αβ unsaturated carbonyl compounds

تعداد نتایج: 252812  

2008
M. A. Azam B. R. P. Kumar S. Shalini B. Suresh T. K. Reddy C. D. Reddy

A number of substituted-α,β-unsaturated carbonyl compounds (1a-i) were prepared by Claisen-Schmidt condensation of substituted acetophenone with selected araldehydes, which on cycloaddition with thiourea furnished 4,6-disubstituted pyrimidine-2-thiols (2a-i). Reaction of (2a-i) with ethyl chloroacetate followed by condensation with hydrazine hydrate yielded 2-[(4,6-disubstituted pyrimidine-2-yl...

Journal: :Journal of Synthetic Organic Chemistry, Japan 1966

2015
Liang Lu Michael J. Meehan Shuo Gu Zhilong Chen Weipeng Zhang Gen Zhang Lingli Liu Xuhui Huang Pieter C. Dorrestein Ying Xu Bradley S. Moore Pei-Yuan Qian

Thalassospiramides comprise a large family of lipopeptide natural products produced by Thalassospira and Tistrella marine bacteria. Here we provide further evidence of their nanomolar inhibitory activity against the human calpain 1 protease. Analysis of structure-activity relationship data supported our hypothesis that the rigid 12-membered ring containing an α,β-unsaturated carbonyl moiety is ...

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