نتایج جستجو برای: 3a5 cpy

تعداد نتایج: 371  

Journal: :Molecular pharmacology 2000
J Marill T Cresteil M Lanotte G G Chabot

Cytochrome P450 (P450)-dependent metabolism of all-trans-retinoic acid (atRA) is important for the expression of its biological activity. Because the human P450s involved in the formation of the principal atRA metabolites have been only partially identified, the purpose of this study was to identify the human P450s involved in atRA metabolism. The use of phenotyped human liver microsomes (n = 1...

2015
Dhanuka P. Wasalathanthri Dandan Li Donghui Song Zhifang Zheng Dharamainder Choudhary Ingela Jansson Xiuling Lu John B. Schenkman James F. Rusling

[Ru(bpy)2(PVP)10] (RuPVP (bpy = 2,2-bipyridyl; PVP = poly(4-vinylpyridine)) was synthesized and characterized as described previously. Styrene (MW= 104.15), 2Acetylaminofluorene (2-AAF, MW= 223.27), 4-(Methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK, MW= 207.23), poly(diallyldimethylammonium chloride) (PDDA, average Mw= 100,000200,000), poly(sodium 4-styrenesulfonate) (PSS, average MW= 70000),...

Journal: :Basic <html_ent glyph="@amp;" ascii="&amp;"/> Clinical Pharmacology <html_ent glyph="@amp;" ascii="&amp;"/> Toxicology 2006

Journal: :Molecular pharmacology 2016
Yanjun Hong Yvonne Mei Fen Chia Ray Hng Yeo Gopalakrishnan Venkatesan Siew Kwan Koh Christina Li Lin Chai Lei Zhou Pipin Kojodjojo Eric Chun Yong Chan

Dronedarone is an antiarrhythmic agent approved in 2009 for the treatment of atrial fibrillation. An in-house preliminary study demonstrated that dronedarone inhibits cytochrome P450 (CYP) 3A4 and 3A5 in a time-dependent manner. This study aimed to investigate the inactivation of CYP450 by dronedarone. We demonstrated for the first time that both dronedarone and its main metabolite N-desbutyl d...

2015
Yanjun Hong Yvonne Mei Fen Chia Ray Hng Yeo Gopalakrishnan Venkatesan Siew Kwan Koh Christina Li Lin Chai Lei Zhou Pipin Kojodjojo Eric Chun Yong Chan

Dronedarone is an antiarrhythmic agent approved in 2009 for the treatment of atrial fibrillation. An in-house preliminary study demonstrated that dronedarone inhibits cytochrome P450 (CYP) 3A4 and 3A5 in a time-dependent manner. This study aimed to investigate the inactivation of CYP450 by dronedarone. We demonstrated for the first time that both dronedarone and its main metabolite N-desbutyl d...

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