نتایج جستجو برای: antileishmanial agent

تعداد نتایج: 254431  

Journal: :International Journal of Biological Macromolecules 2015

2017
Madiha Ahmed Humaira Fatima Muhammad Qasim Bilquees Gul Ihsan-ul-Haq

BACKGROUND Plants have served either as a natural templates for the development of new chemicals or a phytomedicine since antiquity. Therefore, the present study was aimed to appraise the polarity directed antioxidant, cytotoxic, protein kinase inhibitory, antileishmanial and glucose modulatory attributes of a Himalayan medicinal plant- Quercus dilatata. METHODS Total phenolic and flavonoid c...

Journal: :Journal of Enzyme Inhibition and Medicinal Chemistry 2017

Journal: :Journal of Antimicrobial Chemotherapy 2008

Journal: :Memorias do Instituto Oswaldo Cruz 2004
Lianet Monzote Fidalgo Ana Margarita Montalvo Alvarez Lisset Fonseca Geigel Rolando Pérez Pineiro Margarita Suárez Navarro Hortensia Rodríguez Cabrera

Current therapy for leishmaniasis is not satisfactory. We describe the in vitro antiproliferative effects of new thiadiazine derivatives against Leishmania amazonensis. The compounds were found to be active against the amastigote form of the parasite, inhibiting parasite growing, from 10 to 89%, at a concentration of 100 ng/ml. This activity suggests that thiadiazine derivatives could be consid...

2018
Valentin Schatz Patrick Neubert Franz Rieger Jonathan Jantsch

Low oxygen environments and accumulation of hypoxia-inducible factors (HIFs) are features of infected and inflamed tissues. Here, we summarize our current knowledge on oxygen levels found in Leishmania-infected tissues and discuss which mechanisms potentially contribute to local tissue oxygenation in leishmanial lesions. Moreover, we review the role of hypoxia and HIF-1 on innate antileishmania...

2014
Juliana Q. Reimão Danilo C. Miguel Noemi N. Taniwaki Cristiana T. Trinconi Jenicer K. U. Yokoyama-Yasunaka Silvia R. B. Uliana

BACKGROUND The treatment of leishmaniasis relies mostly on parenteral drugs with potentially serious adverse effects. Additionally, parasite resistance in the treatment of leishmaniasis has been demonstrated for the majority of drugs available, making the search for more effective and less toxic drugs and treatment regimens a priority for the control of leishmaniasis. The aims of this study wer...

Journal: :Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 2013
G Morizot E Kendjo O Mouri M Thellier A Pérignon F Foulet F Cordoliani E Bourrat E Laffitte I Alcaraz N Bodak C Ravel M Vray M Grogl D Mazier E Caumes L Lachaud P A Buffet

BACKGROUND Cutaneous leishmaniasis (CL) is a disfiguring but not life-threatening disease. Because antileishmanial drugs are potentially toxic, the World Health Organization (WHO) recommends simple wound care or local therapy as first-line treatment, followed or replaced by systemic therapy if local therapy fails or cannot be performed. METHODS To determine the feasibility and impact of the r...

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