نتایج جستجو برای: atovaquone

تعداد نتایج: 456  

2011
Laurent Dembele Audrey Gego Anne-Marie Zeeman Jean-François Franetich Olivier Silvie Armelle Rametti Roger Le Grand Nathalie Dereuddre-Bosquet Robert Sauerwein Geert-Jan van Gemert Jean-Christophe Vaillant Alan W. Thomas Georges Snounou Clemens H. M. Kocken Dominique Mazier

BACKGROUND Amongst the Plasmodium species in humans, only P. vivax and P. ovale produce latent hepatic stages called hypnozoites, which are responsible for malaria episodes long after a mosquito bite. Relapses contribute to increased morbidity, and complicate malaria elimination programs. A single drug effective against hypnozoites, primaquine, is available, but its deployment is curtailed by i...

2007
Ahmad Saleh Stefan Baumeister Wolfgang Bohne

Both apicomplexan parasites Toxoplasma gondii and Plasmodium falciparum lack type I NADH dehydrogenases (complex I), but instead encode alternative (type II) NADH dehydrogenases, which are absent in mammalian cells and are thus considered as promising antimicrobial drug targets. The quinolone-like compound 1-hydroxy-2-dodecyl-4(1)quinolone (HDQ) was recently 5 described as a high affinity inhib...

Journal: :Archives of internal medicine 2002
Sue J Goldie Jonathan E Kaplan Elena Losina Milton C Weinstein A David Paltiel George R Seage Donald E Craven April D Kimmel Hong Zhang Calvin J Cohen Kenneth A Freedberg

BACKGROUND Human immunodeficiency virus (HIV)-infected patients receiving highly active antiretroviral therapy (HAART) have experienced a dramatic decrease in Pneumocystis carinii pneumonia (PCP), necessitating reassessment of clinical guidelines for prophylaxis. METHODS A simulation model of HIV infection was used to estimate the lifetime costs and quality-adjusted life expectancy (QALE) for...

Journal: :Biochimica et biophysica acta 2007
Jacques J Kessl Nikolai V Moskalev Gordon W Gribble Mohamed Nasr Steven R Meshnick Bernard L Trumpower

Hydroxy-naphthoquinones are competitive inhibitors of the cytochrome bc(1) complex that bind to the ubiquinol oxidation site between cytochrome b and the iron-sulfur protein and presumably mimic a transition state in the ubiquinol oxidation reaction catalyzed by the enzyme. The parameters that affect efficacy of binding of these inhibitors to the bc(1) complex are not well understood. Atovaquon...

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