نتایج جستجو برای: selectivity modeling

تعداد نتایج: 433956  

Journal: :Journal of medicinal chemistry 2009
Chia-Hui Lin Yi-Hui Peng Mohane Selvaraj Coumar Santhosh Kumar Chittimalla Chun-Chen Liao Ping-Chiang Lyn Chin-Chieh Huang Tzu-Wen Lien Wen-Hsing Lin John T-A Hsu Jai-Hong Cheng Xin Chen Jian-Sung Wu Yu-Sheng Chao Hwei-Jen Lee Chiun-Gung Juo Su-Ying Wu Hsing-Pang Hsieh

Utilizing medicinal chemistry design strategies such as benzo splitting and ring expansion, we converted PPARalpha/gamma dual agonist 1 to selective PPARgamma agonists 19 and 20. Compounds 19 and 20 were 2- to 4-fold better than rosiglitazone at PPARgamma receptor, with 80- to 100-fold PPARgamma selectivity over PPARalpha receptor. X-ray cocrystal studies in PPARgamma and modeling studies in PP...

J. Abdi N. M. Mahmoodi

Herein, magnetic cobalt ferrite nanoparticles (CFNPs) was synthesized and its surface was modified by cationic surfactant (cetyltrimethyl ammonium bromide: CTAB) and its potential to selective removal of dye from multicomponent (ternary) system was investigated. Direct red 31 (DR31), Direct green 6 (DG6) and Direct red 23 (DR23) were used as a model dyes. The characteristics of the synthesi...

Journal: :Current Biology 2017
Tirthabir Biswas Chi-Hon Lee

Visual motion detection in insects is mediated by three-input detectors that compare inputs of different spatiotemporal properties. A new modeling study shows that only a small subset of possible arrangements of the input elements provides high direction-selectivity.

2015
Hanchen Xiong Antonio Jose Rodríguez-Sánchez Sándor Szedmák Justus H. Piater

This paper investigates how utilizing diversity priors can discover early visual features that resemble their biological counterparts. The study is mainly motivated by the sparsity and selectivity of activations of visual neurons in area V1. Most previous work on computational modeling emphasizes selectivity or sparsity independently. However, we argue that selectivity and sparsity are just two...

Journal: :iranian journal of pharmaceutical research 0
bo wei lanzhou university of technology zhongduo yang lanzhou university of technology dan-feng shi lanzhou university xiaojun yao lanzhou university minggang wang lanzhou university of technology

seven stilbenes and one catechin were bioactivity-guidedly isolated from the rhizomes of rheum palmatem. their structures were identified as piceatannol(1), resveratrol(2), piceid(3), rhapontigenin(4), piceatannol-3'-o-β-d-glucopyranoside(5), rhaponticin(6), catechin(7) and desoxyrhapontigenin(8). anti-monoamine oxidase (mao) activities of compounds 1–8 were tested. compounds 1 and 8 showe...

Journal: :Neuron 2011
Bao-hua Liu Ya-tang Li Wen-pei Ma Chen-jie Pan Li I. Zhang Huizhong Whit Tao

Orientation selectivity (OS) is an emergent property in the primary visual cortex (V1). How OS arises from synaptic circuits remains unsolved. Here, in vivo whole-cell recordings in the mouse V1 revealed that simple cells received broadly tuned excitation and even more broadly tuned inhibition. Excitation and inhibition shared a similar orientation preference and temporally overlapped substanti...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید