نتایج جستجو برای: 2 methylpropyl ethanoate

تعداد نتایج: 2525279  

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2000
C Teyssier M H Siess

The metabolism of dipropyl disulfide (DPDS), an Allium sulfur compound, was investigated in rat liver cell subfractions and in an isolated perfused rat liver. DPDS is oxidized to dipropyl thiosulfinate (DPDSO) by rat microsomes. The contribution of cytochrome P450 enzymes (CYPs) or flavin-containing monooxygenases (FMO) to the formation of DPDSO from its precursor was investigated. In rat micro...

2016
Yasuhiro Imaeda Hidekazu Tokuhara Yoshiyuki Fukase Ray Kanagawa Yumiko Kajimoto Keiji Kusumoto Mitsuyo Kondo Gyorgy Snell Craig A. Behnke Takanobu Kuroita

The aspartic proteinase renin is an attractive target for the treatment of hypertension and cardiovascular/renal disease such as chronic kidney disease and heart failure. We introduced an S1' site binder into the lead compound 1 guided by structure-based drug design (SBDD), and further optimization of physicochemical properties led to the discovery of benzimidazole derivative 10 (1-(4-methoxybu...

Journal: :Acta Crystallographica Section E Structure Reports Online 2008

Journal: :Journal of neurology, neurosurgery, and psychiatry 1975
D Burke C Hammond N Skuse R F Jones

The efficacy of a selective fusimotor suppressant, the phenothiazine (+/-)-10-3-dimethylamino-2-methylpropyl)-2-valeroylphenothiazine, has been assessed in a double-blind crossover trail in eight patients suffering from cerebral spasticity and one patient suffering from spinal spasticity. Dosage was 40 mg daily. Independent clinical and electromyographic methods of assessment were used. The act...

Journal: :Acta Crystallographica Section E Structure Reports Online 2011

Journal: :Acta Crystallographica Section E Structure Reports Online 2008

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