نتایج جستجو برای: antimony compounds

تعداد نتایج: 230084  

Journal: :Journal of Applied Animal Research 1996

2018
Lucas S Magalhães Lays GS Bomfim Sthefanne G Mota Geydson S Cruz Cristiane B Corrêa Diego M Tanajura Michael W Lipscomb Valéria M Borges Amélia R de Jesus Roque P de Almeida Tatiana R de Moura

BACKGROUND Treatment-refractory visceral leishmaniasis (VL) has become an important problem in many countries. OBJECTIVES We evaluated the antimony-resistance mechanisms of Leishmania infantum isolated from VL patients refractory or responsive to treatment with pentavalent antimony. METHODS Strains isolated from antimony-refractory patients (in vitro antimony-resistant isolates) and antimony-re...

Journal: :Antimicrobial agents and chemotherapy 1997
M Ephros E Waldman D Zilberstein

An axenic amastigote culture system was utilized to directly assess the stage-specific antileishmanial effects of antimony on amastigotes of Leishmania donovani devoid of the macrophage host cell. Pentostam, which contains antimony in the form of sodium stibogluconate and the preservative chlorocresol, was used. Cell density was quantified by measuring the activity of the stable enzyme ornithin...

2013
Marcele Neves Rocha Paula Monalisa Nogueira Cynthia Demicheli Ludmila Gonçalvez de Oliveira Meiriane Mariano da Silva Frédéric Frézard Maria Norma Melo Rodrigo Pedro Soares

Leishmania amazonensis is the etiologic agent of the cutaneous and diffuse leishmaniasis often associated with drug resistance. Lapachol [2-hydroxy-3-(3'-methyl-2-butenyl)-1,4-naphthoquinone] displays a wide range of antimicrobial properties against many pathogens. In this study, using the classic microscopic in vitro model, we have analyzed the effects of a series of lapachol and chlorides com...

Journal: :research in pharmaceutical sciences 0

the six elements commonly known as metalloids are boron, silicon, germanium, arsenic, antimony, and tellurium. metalloid containing compounds have been used as antiprotozoal drugs. boron-based drugs, the benzoxaboroles have been exploited as potential treatments for neglected tropical diseases. arsenic has been used as a medicinal agent and arsphenamine was the main drug used to treat syphilis....

Journal: :Antimicrobial agents and chemotherapy 2005
André Gustavo Tempone Ana Cláudia Melo Pompeu da Silva Carlos Alberto Brandt Fernanda Scalzaretto Martinez Samanta Etel Treiger Borborema Maria Amélia Barata da Silveira Heitor Franco de Andrade

The antileishmanial efficacy of four novel quinoline derivatives was determined in vitro against Leishmania chagasi, using extracellular and intracellular parasite models. When tested against L. chagasi-infected macrophages, compound 3b demonstrated 8.3-fold greater activity than did the standard pentavalent antimony. No significant activity was found for compounds 3a, 4a, and 4b. The antilesih...

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