نتایج جستجو برای: benzimidazolone

تعداد نتایج: 55  

Journal: :The Journal of pharmacology and experimental therapeutics 2000
A K Singh D C Devor A C Gerlach M Gondor J M Pilewski R J Bridges

We previously demonstrated that 1-ethyl-2-benzimidazolone (1-EBIO) directly activates basolateral membrane calcium-activated K(+) channels (K(Ca)), thereby stimulating Cl(-) secretion across several epithelia. In our pursuit to identify potent modulators of Cl(-) secretion that may be useful to overcome the Cl(-) secretory defect in cystic fibrosis (CF), we have identified chlorzoxazone [5-chlo...

2011
Eva K. Roth Stephanie Hirtz Julia Duerr Daniel Wenning Irmgard Eichler Hans H. Seydewitz Margarida D. Amaral Marcus A. Mall

BACKGROUND The identification of strategies to improve mutant CFTR function remains a key priority in the development of new treatments for cystic fibrosis (CF). Previous studies demonstrated that the K⁺ channel opener 1-ethyl-2-benzimidazolone (1-EBIO) potentiates CFTR-mediated Cl⁻ secretion in cultured cells and mouse colon. However, the effects of 1-EBIO on wild-type and mutant CFTR function...

Abdelkader Zarrouk, Abdeslam El Assyry Bouziane Benali Brahim Lakhrissi Fouad Benhiba Fouad Bentiss Hassan Rabaâ Ismail Warad M'Hamed Touil

The adsorption behavior of Benzimidazol-2-one (Bz), 5-Methylbenzimidazol-2-one(CH3Bz) and 5-Chlorobenzimidazol-2-one (ClBz) as inhibitors for mild steel corrosion in HCl 1M have been studied computationally using density functional theory (DFT) calculations with the hybrid B3LYP functional. The calculations were focused on the protonated forms of the molecules under study, seeing tha...

2001
Thomas H. Fife

p-Nitrophenyl N-(2-mercaptophenyl)-N-methylcarbamate cyclizes rapidly at 25' to N-methylbenzothiazolone with release of p-nitrophenol. The pH-rate constant profile is sigmoidal with pK,,, = 8.7. The effective molarity of the neighboring sulfhydryl group is 1.4 X los M in comparison with bimolecular attack of thiols on p-nitrophenyl N-methyl-Nphenylcarbamate. The pH-rate constant profile for cyc...

2014
Jian Lü Cristina Perez-Krap Mikhail Suyetin Nada H. Alsmail Yong Yan Sihai Yang William Lewis Elena Bichoutskaia Chiu C. Tang Alexander J. Blake Rong Cao Martin Schröder

A robust binary hydrogen-bonded supramolecular organic framework (SOF-7) has been synthesized by solvothermal reaction of 1,4-bis-(4-(3,5-dicyano2,6-dipyridyl)dihydropyridyl)benzene (1) and 5,5′-bis(azanediyl)-oxalyl-diisophthalic acid (2). Single crystal Xray diffraction analysis shows that SOF-7 comprises 2 and 1,4-bis-(4-(3,5-dicyano-2,6-dipyridyl)pyridyl)benzene (3); the latter formed in si...

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