A novel series of various 2-hydroxypyrrolidine/piperidine derivatives were synthesized and their antibacterial activity against MTCC bacterial strains, anticancer activity and larvicidal effects were studied. Among the ten synthesized compounds, three were found to be antibacterial in nature. All the five test strains were highly sensitive to 1-(quinolin-3-yl) pyrrolidin-2-ol (P7), moderately s...

A novel series of glucosyl thioureas were synthesized in good overall yields (up to 37% over four steps) from d-glucose and primary amines, and their larvicidal activities toward Mythimna separata Walker were also investigated. This new class of glucosyl thioureas demonstrated low to moderate growth inhibition activity of Mythiman separata Walker, with a growth inhibitory rate of up to 47.5% at...

This study investigated the biological activities of five benthic marine algae collected from Northeastern Region of Brazil. The tested activities included larvicidal activity against Aedes aegypti, molluscicidal activity against Biomphalaria glabrata, and toxicity against Artemia salina. Extracts of Ulva lactuca (Chlorophyta), Padina gymnospora, Sargassum vulgare (Phaeophyta), Hypnea musciform...

BACKGROUND Aedes aegypti L. is the major vector of dengue fever and dengue hemorrhagic fever. In an effort to find effective tools for control programs to reduce mosquito populations, the authors assessed the acute toxicities of 14 monoterpenoids, trans-anithole and the essential oil of rosemary against different larval stages of Ae. aegypti. The potential for piperonyl butoxide (PBO) to act as...

In order to identify novel chlorantraniliprole derivatives as potential insecticides or fungicides, 25 analogues of chlorantraniliprole were synthesized. The insecticidal activities against oriental armyworm and the antifungal activities against five typical fungi of these derivatives were tested. Compounds 2u, 2x and 2y exhibited good activities against oriental armyworm, especially compounds ...

background: plant extracts and oils may act as alternatives to conventional pesticides for malaria vector control. the aim of this study was to evaluate the larvicidal activity of essential oils of three plants of apiaceae family against anophe­les stephensi , the main malaria vector in iran. methods: essential oils from heracleum persicum , foeniculum vulgare and coriandrum sativum seeds were ...

The present study aims to investigate the larvicidal activity of essential oils rhizomes Zingiber officinalis, leaves Tithonia diversifolia and Bidens pilosa on mature immature larvae Anopheles gambiae s.l. chemical composition was determined by Gas Chromatography (GC) Mass Spectrometry (GC/MS) coupling. activities against An. monitored in laboratory using world health organisation protocol. Ch...

Mangostin derived from mangosteen was identiÞed as a mosquito sterol carrier protein-2 inhibitor via high throughput insecticide screening. -Mangostin was tested for its larvicidal activity against third instar larvae of six mosquito species, and the median lethal concentration values range from 0.84 to 2.90 ppm. The residual larvicidal activity of -mangostin was examined under semiÞeld conditi...

BACKGROUND Taking into account the improvement in insecticidal activity by the inclusion of fluorine in the hydrazone moiety, the authors synthesized new 4-fluorobenzoic acid hydrazides and 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazoles, substituting a phenyl group or a heteroaryl ring carrying one or two atoms of F, Cl and Br, and investigated their biting deterrent and larvicidal ac...