نتایج جستجو برای:

تعداد نتایج: 4491  

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2017
Amy Walz Andrey Ugolkov Sunandana Chandra Alan Kozikowski Benedito A Carneiro Thomas V O'Halloran Francis J Giles Daniel D Billadeau Andrew P Mazar

Glycogen synthase kinase-3β (GSK-3β), a serine/threonine protein kinase, is a complex regulator of numerous cellular functions. GSK-3β is a unique kinase which is constitutively active in resting and nonstimulated cells. GSK-3β has been implicated in a wide range of diseases including neurodegeneration, inflammation and fibrosis, noninsulin-dependent diabetes mellitus, and cancer. It is a regul...

Journal: :Oxidative medicine and cellular longevity 2016
Yuanyuan Cheng Zhengyuan Xia Yifan Han Jianhui Rong

The opening of mitochondrial permeability transition pore (mPTP) is a major cause of cell death in ischemia reperfusion injury. Based on our pilot experiments, plant natural product formononetin enhanced the survival of rat cardiomyocyte H9c2 cells during oxygen glucose deprivation (OGD) and reoxygenation. For mechanistic studies, we focused on two major cellular factors, namely, reactive oxyge...

Journal: :Molecular bioSystems 2013
Vatsala Malik Meng Zhang Lynn G Dover Julian S Northen Anthony Flinn Justin J Perry Gary W Black

The main objectives of this work were to characterise a range of purified recombinant sterol 3β-glucosyltransferases and show that rational sampling of the diversity that exists within sterol 3β-glucosyltransferase sequence space can result in a range of enzyme selectivities. In our study the catalytically active domain of the Saccharomyces cerevisiae 3β-glucosyltransferase was used to mine put...

Journal: :International journal of molecular medicine 2015
Yichao Yan Guangying Li Xiaofeng Tian Yingjiang Ye Zhidong Gao Jihong Yao Feng Zhang Shan Wang

Ischemic preconditioning (IPC) ameliorates ischemia/reperfusion (I/R) injury in a number of organs, and the glycogen synthase kinase-3β (GSK-3β)/β-catenin signaling pathway regulates I/R-induced proliferation and apoptosis in the central nervous system and heart. However, the function of this signaling pathway in IPC during liver I/R remains unclear. Thus, in this study, we aimed to investigte ...

Journal: :The Journal of clinical investigation 2014
Spyridon Theofilopoulos William J Griffiths Peter J Crick Shanzheng Yang Anna Meljon Michael Ogundare Satish Srinivas Kitambi Andrew Lockhart Karin Tuschl Peter T Clayton Andrew A Morris Adelaida Martinez M Ashwin Reddy Andrea Martinuzzi Maria T Bassi Akira Honda Tatsuki Mizuochi Akihiko Kimura Hiroshi Nittono Giuseppe De Michele Rosa Carbone Chiara Criscuolo Joyce L Yau Jonathan R Seckl Rebecca Schüle Ludger Schöls Andreas W Sailer Jens Kuhle Matthew J Fraidakis Jan-Åke Gustafsson Knut R Steffensen Ingemar Björkhem Patrik Ernfors Jan Sjövall Ernest Arenas Yuqin Wang

Cholestenoic acids are formed as intermediates in metabolism of cholesterol to bile acids, and the biosynthetic enzymes that generate cholestenoic acids are expressed in the mammalian CNS. Here, we evaluated the cholestenoic acid profile of mammalian cerebrospinal fluid (CSF) and determined that specific cholestenoic acids activate the liver X receptors (LXRs), enhance islet-1 expression in zeb...

2014
Hui Zhang Wenjie Wang Haoshu Fang Yan Yang Xiaolan Li Junli He Xiaojing Jiang Weipeng Wang Shenpei Liu Jifa Hu Anding Liu Uta Dahmen Olaf Dirsch

Liver dysfunction has been known to occur frequently in cases of sepsis. Excessive inflammation and apoptosis are pathological features of acute liver failure. Recent studies suggest that activation of glycogen synthase kinase- (GSK-) 3β is involved in inflammation and apoptosis. We aimed to investigate the protective effects of GSK-3β inhibition on polymicrobial sepsis-induced liver injury and...

2015
Xian Li Yimin Jia Runsheng Li Zhiyuan Sun Xi Li Shiyan Sui Ruqian Zhao

BACKGROUND Hepatic 3β-hydroxysteroid dehydrogenase (3β-HSD) plays an important role in steroid inactivation and catabolism. Serum concentrations of steroid hormones differ significantly between breeds in pigs, however the molecular mechanism regulating hepatic 3β-HSD expression in different breeds of pigs is poorly understood. In the present study, we used preweaning purebred male Large White (...

2016
Toru Hanamura Tokiko Ito Toshiharu Kanai Kazuma Maeno Yasuyo Shimojo Takeshi Uehara Takashi Suzuki Shin‐ichi Hayashi Ken‐ichi Ito

Active sex steroids including estrogens and androgens are locally produced from circulating inactive steroids by various steroid-metabolizing enzymes, and play pivotal roles in the progression of hormone-dependent breast cancers. Human 3β-hydroxysteroid dehydrogenase type 1 (3β-HSD type 1) is a critical enzyme in the formation of all classes of active steroid hormones, and is also involved in t...

2013
Martin Krøyer Rasmussen Bo Ekstrand Galia Zamaratskaia

This review focuses on the expression and regulation of 3β-hydroxysteroid dehydrogenase/Δ⁵-Δ⁴ isomerase (3β-HSD), with emphasis on the porcine version. 3β-HSD is often associated with steroidogenesis, but its function in the metabolism of both steroids and xenobiotics is more obscure. Based on currently available literature covering humans, rodents and pigs, this review provides an overview of ...

Journal: :Frontiers in veterinary science 2014
Michael H. Kogut Christina L. Swaggerty Hsin-I Chiang Kenneth J. Genovese Haiqi He Huaijun Zhou Ryan J. Arsenault

A microarray-assisted gene expression screen of chicken heterophils revealed glycogen synthase kinase-3β (GSK-3β), a multifunctional Ser/Thr kinase, to be consistently upregulated 30-180 min following stimulation with Salmonella enterica serovar Enteritidis (S. Enteritidis). The present study was designed to delineate the role of GSK-3β in regulating the innate function of chicken heterophils i...

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