نتایج جستجو برای: acetylcholinesterase inhibitors

تعداد نتایج: 194637  

Journal: :Molecules 2016
Youssef Dgachi Oscar M Bautista-Aguilera Mohamed Benchekroun Hélène Martin Alexandre Bonet Damijan Knez Justyna Godyń Barbara Malawska Stanislav Gobec Mourad Chioua Jana Janockova Ondrej Soukup Fakher Chabchoub José Marco-Contelles Lhassane Ismaili

We report herein the straightforward two-step synthesis and biological assessment of novel racemic benzochromenopyrimidinones as non-hepatotoxic, acetylcholinesterase inhibitors with antioxidative properties. Among them, compound 3Bb displayed a mixed-type inhibition of human acetylcholinesterase (IC50 = 1.28 ± 0.03 μM), good antioxidant activity, and also proved to be non-hepatotoxic on human ...

Amna Saeed Aziz-ur Rehman Khalid Mohmmed Khan Muhammad Abbasi, Muhammad Ashraf, Syeda Abida Ejaz

The present study reports the synthesis of a series N-substituted derivatives of brominated 2-phenitidine. First, the reaction of 2-phenitidine (1) with benzenesulfonyl chloride (2) in aqueous media yielded N-(2-ethoxyphenyl) benzenesulfonamide (3), which was then subjected to bromination with bromine in the presence of glacial acetic acid to give N-(4,5-dibromo-2-ethoxyphenyl)benzenesulfonamid...

Journal: :Drug Designing & Intellectual Properties International Journal 2018

Journal: :Psychiatria Danubina 2009
Ninoslav Mimica Paola Presecki

The aim of this review is to describe side effects of five antidementives which are approved by the United States Food and Drug Administration (FDA); four acetylcholinesterase inhibitors and one glutamate - or N-metyl-D-aspartat receptor antagonist - memantine. The antidementives are well tolerated and undesired effects are rare; except hepatotoxicity of tacrine and gastrointestinal side effect...

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