نتایج جستجو برای: cholesteryl ester transfer protein cetp gene

تعداد نتایج: 2254676  

Journal: :Journal of lipid research 2010
Mollie Ranalletta Kathleen K Bierilo Ying Chen Denise Milot Qing Chen Elaine Tung Caroline Houde Nadine H Elowe Margarita Garcia-Calvo Gene Porter Suzanne Eveland Betsy Frantz-Wattley Mike Kavana George Addona Peter Sinclair Carl Sparrow Edward A O'Neill Ken S Koblan Ayesha Sitlani Brian Hubbard Timothy S Fisher

Cholesteryl ester transfer protein (CETP) has been identified as a novel target for increasing HDL cholesterol levels. In this report, we describe the biochemical characterization of anacetrapib, a potent inhibitor of CETP. To better understand the mechanism by which anacetrapib inhibits CETP activity, its biochemical properties were compared with CETP inhibitors from distinct structural classe...

2015
Shinji Yokoyama Kuniko Okumura-Noji Rui Lu

Schistosoma japonicum, once endemic all the East Asia, remains as a serious public health problem in certain regions. Ectopic egg embryonation in the liver causes granulomatosis and eventually fatal cirrhosis, so that prevention of this process is one of the keys to reduce its mortality. The embryonation requires cholesteryl ester from HDL of the host blood for egg yolk formation, and this reac...

Journal: :Journal of lipid research 2010
Silvia Bijland Sjoerd A A van den Berg Peter J Voshol Anita M van den Hoek Hans M G Princen Louis M Havekes Patrick C N Rensen Ko Willems van Dijk

The cholesteryl ester transfer protein (CETP) facilitates the bidirectional transfer of cholesteryl esters and triglycerides (TG) between HDL and (V)LDL. By shifting cholesterol in plasma from HDL to (V)LDL in exchange for VLDL-TG, CETP aggravates atherosclerosis in hyperlipidemic APOE*3-Leiden (E3L) mice. The aim of this study was to investigate the role of CETP in TG metabolism and high-fat d...

2002
James B. Moberly Mark J. Bamberger

Sensitive immunoradiometric (IRMA) and ELISA Supplementary key words sandwich blotting immunoblotting assays for cholesteryl ester transfer protein (CETP) have been native gel electrophoresis prebeta migrating Superose Superdex developed using two different monoclonal antibodies (MAbs). HepG2 cells The MAbs were prepared against human plasma CETP and demonstrated specificity by their inhibition...

Journal: :Aging cell 2012
Lei Yu Joshua M Shulman Lori Chibnik Sue Leurgans Julie A Schneider Philip L De Jager David A Bennett

The cholesteryl ester transfer protein (CETP) gene plays an essential role in regulating cholesterol homeostasis and is a candidate susceptibility gene for late-onset Alzheimer's disease (AD). Recent finding suggests that the CETP I405V polymorphism (rs5882) is associated with a slower rate of memory decline and a lower risk of incident dementia. Using data from two ongoing epidemiologic clinic...

Journal: :Journal of lipid research 2001
Y Fusegawa K L Kelley J K Sawyer R N Shah L L Rudel

CETP activity, measured as transfer of cholesteryl ester from exogenous HDL to exogenous VLDL and LDL, reflecting CETP mass as determined by ELISA, was documented in three groups of St. Kitts vervet monkeys fed diets enriched in saturated (Sat), monounsaturated (Mono), or n-6 polyunsaturated (Poly) fatty acids. CETP activity was not different when comparing the three dietary fats. However, CETP...

Journal: :Journal of lipid research 2003
Richard E Morton Diane J Greene

Cholesteryl ester transfer protein (CETP) activity is regulated, in part, by lipoprotein composition. We previously demonstrated that CETP activity follows saturation kinetics as cholesteryl ester (CE) levels in the phospholipid surface of donor particles are increased. We propose here that the plateau of CETP activity occurs because the surface concentration of CE in the acceptor becomes rate ...

Journal: :The Journal of biological chemistry 2000
T Gautier D Masson J P de Barros A Athias P Gambert D Aunis M H Metz-Boutigue L Lagrost

The aim of the present study was to identify the protein that accounts for the cholesteryl ester transfer protein (CETP)-inhibitory activity that is specifically associated with human plasma high density lipoproteins (HDL). To this end, human HDL apolipoproteins were fractionated by preparative polyacrylamide gradient gel electrophoresis, and 30 distinct protein fractions with molecular masses ...

Journal: :Molecules 2017
Xinran Wang Xuehua Lin Xuanqi Xu Wei Li Lijuan Hao Chunchi Liu Dongmei Zhao Maosheng Cheng

Cholesteryl ester transfer protein (CETP) has been identified as a potential target for cardiovascular disease (CVD) for its important role in the reverse cholesteryl transfer (RCT) process. In our previous work, compound 5 was discovered as a moderate CETP inhibitor. The replacement of the amide linker by heterocyclic aromatics and then a series of N,N-substituted-4-arylthiazole-2-methylamine ...

Journal: :Arteriosclerosis and thrombosis : a journal of vascular biology 1994
T Arai S Yamashita K Hirano N Sakai K Kotani S Fujioka S Nozaki Y Keno M Yamane E Shinohara

It is well known that obesity is frequently associated with low levels of serum high-density lipoprotein (HDL) cholesterol. However, the mechanism for this reduction has not been fully clarified. Cholesteryl ester transfer protein (CETP) transfers cholesteryl ester from HDL to apolipoprotein B-containing lipoproteins and plays an important role in regulating the concentration and composition of...

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