نتایج جستجو برای: fingolimod fty720

تعداد نتایج: 1720  

2015
Jens Kuhle Giulio Disanto Johannes Lorscheider Tracy Stites Yu Chen Frank Dahlke Gordon Francis Anupama Shrinivasan Ernst-Wilhelm Radue Gavin Giovannoni Ludwig Kappos

OBJECTIVE We assessed CSF levels of the light chain subunit of neurofilaments (NfL) at baseline and after fingolimod therapy or placebo in patients with relapsing-remitting multiple sclerosis (RRMS). Changes in NfL levels were also correlated with relapse and MRI outcomes. METHODS CSF samples were available, at baseline and 12 months after treatment initiation, from a subset of 36 patients wi...

2016
David C. Miller Karen B. Whittington David D. Brand Karen A. Hasty Edward F. Rosloniec

BACKGROUND Fingolimod (FTY720) is an immunomodulating drug that inhibits sphingosine-1-phosphate binding and blocks T-cell egress from lymph nodes. We analyzed the effect of FTY720 on the autoimmune T- and B-cell response in autoimmune arthritis and studied the mechanisms by which it alters the function of T cells. METHODS Human leukocyte antigen (HLA)-DR1 humanized mice were immunized with t...

2016
Guadalupe Vidal-Martínez Javier Vargas-Medrano Carolina Gil-Tommee David Medina Nathan T. Garza Barbara Yang Ismael Segura-Ulate Samantha J. Dominguez Ruth G. Perez

Patients with Parkinson's disease (PD) often have aggregated α-synuclein (aSyn) in enteric nervous system (ENS) neurons, which may be associated with the development of constipation. This occurs well before the onset of classic PD motor symptoms. We previously found that aging A53T transgenic (Tg) mice closely model PD-like ENS aSyn pathology, making them appropriate for testing potential PD th...

Journal: :Chemistry & biology 2012
Jean Quancard Birgit Bollbuck Philipp Janser Daniela Angst Frédéric Berst Peter Buehlmayer Markus Streiff Christian Beerli Volker Brinkmann Danilo Guerini Paul A Smith Timothy J Seabrook Martin Traebert Klaus Seuwen René Hersperger Christian Bruns Frédéric Bassilana Marc Bigaud

Lymphocyte trafficking is critically regulated by the Sphingosine 1-phosphate receptor-1 (S1P(1)), a G protein-coupled receptor that has been highlighted as a promising therapeutic target in autoimmunity. Fingolimod (FTY720, Gilenya) is a S1P(1) receptor agonist that has recently been approved for the treatment of multiple sclerosis (MS). Here, we report the discovery of NIBR-0213, a potent and...

Journal: :Journal of Pharmacology and Pharmacotherapeutics 2011

2015
A. Leo R. Citraro S. Chimirri F. Scicchitano G. De Sarro E. Russo

Fingolimod (FTY720), a sphingosine-1-phosphate receptor (S1PR) modulator, was the first oral therapy approved by US Food and Drug Administration (FDA) and European Medicines Agency (EMA) for the treatment of relapsing-remitting multiple sclerosis[1]. To date, fingolimod has not been studied in epilepsy models; however, a recent study performed in the lithium-pilocarpine rat model of SE (status ...

Journal: :The Journal of neuroscience : the official journal of the Society for Neuroscience 2014
Dianer Yang Yu-Yo Sun Siddhartha Kumar Bhaumik Yikun Li Jessica M Baumann Xiaoyi Lin Yujin Zhang Shang-Hsuan Lin R Scott Dunn Chia-Yang Liu Feng-Shiun Shie Yi-Hsuan Lee Marsha Wills-Karp Claire A Chougnet Suhas G Kallapur Ian P Lewkowich Diana M Lindquist Kaja Murali-Krishna Chia-Yi Kuan

Intrauterine infection (chorioamnionitis) aggravates neonatal hypoxic-ischemic (HI) brain injury, but the mechanisms linking systemic inflammation to the CNS damage remain uncertain. Here we report evidence for brain influx of T-helper 17 (TH17)-like lymphocytes to coordinate neuroinflammatory responses in lipopolysaccharide (LPS)-sensitized HI injury in neonates. We found that both infants wit...

2015
Jorge Correale Jose Flores Juan Garcia Bonitto Claudia Cárcamo Rodríguez Enedina M. L. Oliveira

UNLABELLED Once-daily fingolimod 0.5 mg (FTY720; Gilenya(®), Novartis Pharma AG, Basel, Switzerland) is a sphingosine 1-phosphate receptor modulator that is approved for the treatment of relapsing multiple sclerosis (MS); currently, this includes approval in 13 Latin American countries. However, despite a well-characterized efficacy and safety profile in a large clinical development program, th...

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