نتایج جستجو برای: propargylamine

تعداد نتایج: 73  

2018
Robby Vroemans Fante Bamba Jonas Winters Joice Thomas Jeroen Jacobs Luc Van Meervelt Jubi John Wim Dehaen

A practical three-step protocol for the assembly of triazolobenzodiazepine-fused diketopiperazines and hydantoins has been developed. The synthesis of these tetracyclic ring systems was initiated by an Ugi reaction, which brought together all necessary functionalities for further transformations. The Ugi adducts were then subjected to a base-induced ring closing and an intramolecular azide-alky...

2012
Hannah K. Murnen Alexei R. Khokhlov Pavel G. Khalatur Rachel A. Segalman Ronald N. Zuckermann

Understanding the driving forces for the collapse of a polymer chain from a random coil to a globule would be invaluable in enabling scientists to predict the folding of polypeptide sequences into defined tertiary structures. The HP model considers hydrophobic collapse to be the major driving force for protein folding. However, due to the inherent presence of chirality and hydrogen bonding in p...

2012
Julie A. Pollock Michelle D. Larrea Jeff S. Jasper Donald P. McDonnell Dewey G. McCafferty

Lysine specific demethylase 1 (LSD1, also known as KDM1) is a histone modifying enzyme that regulates the expression of many genes important in cancer progression and proliferation. It is present in various transcriptional complexes including those containing the estrogen receptor (ER). Indeed, inhibition of LSD1 activity and or expression has been shown to attenuate estrogen signaling in breas...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید