Let n < 0 be arbitrary. A central problem in Euclidean Lie theory is the computation of ideals. We show that ξ ≡ R(∆). Unfortunately, we cannot assume that R̂ ( 1 U , 1 2 ) = { 1 s : r̄−1 (1 ∧ |r̂|) > sin−1 ( β(O) ) sinh−1 (C′−1) } ≥ { Ȳ · 0: αα,F ( ∞−6, . . . , ξ−2 ) < 1 s(y) × log (e± δq) }

In the present work, we report the synthesis and in vitro anticancer and antimicrobial activity evaluation of a new series of 1-substituted-β-carboline derivatives bearing a 4-benzylidene-4H-oxazol-5-one unity at C-3. The compound 2-[1-(4-methoxyphenyl)-9H-β-carbolin-3-yl]-4-(benzylidene)-4H-oxazol-5-one (11) was the most active derivative, exhibiting a potent cytotoxic activity against glioma ...

In order to overcome the rapid biliary excretion of chartreusin, which diminished its activity when administered iv, a series of 3',4'-O-substituted derivatives of chartreusin were synthesized. Exo-type of 3',4'-O-benzylidene-chartreusin was found active both by ip and iv administration. Therefore, this compound was selected for further modification on its 6-phenol to obtain broader spectra and...

The synthesis and evaluation of the anticancer activity of 3'-aryl-5'-arylidene-spiro[3H-indole-3,2'-thiazolidine]-2,4'(1H)-diones and spiro[3H-indole-3,2'-thi-azolidine]-2,4'(1H)-dione-3'-alkanoic acid esters were described. The structure of the compounds was determined by (1)H and (13)C NMR and their in vitro anticancer activity was tested in the National Cancer Institute. Among the tested co...

a number of 6-hydroxy-2-benzylidene-3-coumaranones were synthesized from condensation of 6-hydroxy-3-coumaranone with appropriate aldehydes and were evaluated for their antioxidant activities. the antioxidant activity was assessed using two methods, including, 1,1-biphenyl-2-picrylhydrazyl (dpph) radical scavenging, and reducing power assays. some of the benzylidene coumaranones showed antioxid...

Several 4-arylidene-2-phenyl-1-(2,4,5-trichlorophenyl)-1H-imidazol-5(4H)-ones (4a-q), N-(4-benzylidene-5-oxo-2-phenyl-4,5-dihydroimidazol-1-yl)-4-chlorobenzamides (5a-o) and N-(4-benzylidene-5-oxo-2-phenyl-4,5-dihydroimidazol-1-yl)-2,4-dichlorobenzamides (6a-m) were prepared. All newly synthesized compounds have been tested for their antibacterial activity against gram (+)ve and gram (-)ve bact...

The inhibiting effects of some newly synthesized Schiff bases on the corrosion of Al-Pure in 1.0 M HCl have been studied by means of the chemical and electrochemical methods. The Schiff bases m-Chloroaniline-N-benzylidene (m-CANB), p-Chloroaniline–N-benzylidene (p-CANB), Benzylamine-N-(p-methoxy benzylidene) (BANPMB) and 2-Phenylethylamine-N-(p-methoxy benzylidene) (2PANPMB) were synthesized fr...

A series of 5-benzylidenerhodanine-3-acetamides bearing morpholino-, 4-arylpiperazinyl-, or 4-benzylpiperidinyl- moieties were synthesized and their inhibitory activities against acetylcholinesterase (AChE) were evaluated. Alteration of amide part and substitution on the benzylidene moiety resulted in change of anti-AChE activity. The most active compound was the 1-benzylpiperidinyl derivative ...

Kinetics of the reactions of four benzenesulfonyl-stabilized carbanions (1a-d)- with reference electrophiles (quinone methides 2 and diarylcarbenium ions 3) have been determined in dimethyl sulfoxide solution at 20 degrees C in order to derive the reactivity parameters N and s according to the linear free-energy relationship logk(20 degrees C) = s(N + E) (eqn (1)). The additions of (1a-d)- to o...