نتایج جستجو برای: acid amide hydrolase

تعداد نتایج: 772887  

2008
K. BREDDAM

Treatment of carboxypeptidase Y with ~4C-iodoacetamide caused a drastic reduction in the peptidase activity towards FA-Phe-$Leu-OH while the esterase activity towards FA-Phe 89 the amidase activity towards FA-PhelNH2 and the peptidyl amino acid amide hydrolase activity towards FA-Phe-$GIy-NH2 were much less affected. The loss of peptidase activity could be correlated with the incorporation of a...

Journal: :Journal of Cerebral Blood Flow & Metabolism 2016

Journal: :Bioorganic & medicinal chemistry letters 2008
Ian M Slaymaker Michael Bracey Mauro Mileni Joie Garfunkle Benjamin F Cravatt Dale L Boger Raymond C Stevens

The melting curves of fatty acid amide hydrolase (FAAH) in the presence of 29 reversible inhibitors were measured using a thiol-reactive fluorophore. The thermal stability (T(m)) of the FAAH/inhibitor complex varied significantly depending on the chemical characteristics of the inhibitors, notably variations in the head group. Two separate distributions were observed when T(m) was plotted again...

Journal: :Anesthesiology 2006
Gustav Schelling Daniela Hauer Shahnaz Christina Azad Martin Schmoelz Alexander Chouker Michael Schmidt Cyrill Hornuss Markus Rippberger Josef Briegel Manfred Thiel Michael Vogeser

BACKGROUND The endocannabinoid system includes G-protein-coupled cannabinoid receptors, the endocannabinoids N-arachidonoylethanolamine (anandamide) and 2-arachidonoylglycerol, and multiple enzymes involved in the biosynthesis and degradation of endocannabinoids, including the anandamide metabolizing enzyme fatty acid amide hydrolase. Endocannabinoids play an important role in the physiologic c...

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