نتایج جستجو برای: adrenoceptor antagonists

تعداد نتایج: 56535  

Journal: :The Journal of pharmacology and experimental therapeutics 2014
Mónica Moreira-Rodrigues Ana L Graça Marlene Ferreira Joana Afonso Paula Serrão Manuela Morato Fátima Ferreirinha Paulo Correia-de-Sá Steven N Ebert Daniel Moura

It has been suggested that there is a link between epinephrine synthesis and the development of β2-adrenoceptor-mediated effects, but it remains to be determined whether this development is triggered by epinephrine. The aim of this study was to characterize β-adrenoceptor-mediated relaxation and facilitation of norepinephrine release in the aorta of phenylethanolamine-N-methyltransferase-knocko...

2014
Mónica Moreira-Rodrigues Ana L. Graça Marlene Ferreira Joana Afonso Paula Serrão Manuela Morato Fátima Ferreirinha Paulo Correia-de-Sá Steven N. Ebert Daniel Moura

It has been suggested that there is a link between epinephrine synthesis and the development of b2-adrenoceptor–mediated effects, but it remains to be determined whether this development is triggered by epinephrine. The aim of this study was to characterize b-adrenoceptor–mediated relaxation and facilitation of norepinephrine release in the aorta of phenylethanolamine-Nmethyltransferase–knockou...

Journal: :Circulation research 1986
F M Tayo R D Bevan J A Bevan

The pharmacological characteristics of the postjunctional alpha-adrenoceptors of vascular smooth muscle were studied in ring segments of thoracic aorta, superior mesenteric, and central ear arteries of 4- and 8-week-old, and young adult (12- to 16-week-old) rabbits. Norepinephrine (alpha 1, alpha 2-agonist), phenylephrine (alpha 1-agonist), and UK 14,304-18 (alpha 1-agonist) caused a concentrat...

2000
Gerhard J. Molderings Heinz Bönisch Michael Brüss James Likungu Manfred Göthert

On the basis of data obtained in rabbits, the imidazoline receptor ligand rilmenidine has been suggested to decrease blood pressure in humans by activating central a2A-adrenoceptors. A prerequisite for this hypothesis was the unproved assumption that rabbit and human a2A-adrenoceptors are equally activated by rilmenidine. Because a2A-adrenoceptors in the brain and on cardiovascular sympathetic ...

2006
Tomonori Yamanishi Takao Kamai Ryuji Sakakibara Tomoyuki Uchiyama Tatsuya Yamamoto Takashi Ito Ken-ichiro Yoshida

For the pharmacological treatment of frequency, urgency and/or urge incontinence due to bladder overactivity, anticholinergics have been used as first-choice drugs. However, these drugs can exert severe side effects (accommodation paralysis, constipation, tachycardia, dry mouth and blurred vision) and some patients are refractory to their actions. Thus there is a need for new drug therapies wit...

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