Asymmetric Synthesis of 2,4,5-Trisubstituted Δ2-Thiazolines

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Asymmetric Synthesis of 2,4,5-Trisubstituted Δ2-Thiazolines

Δ(2)-Thiazolines are interesting heterocycles that display a wide variety of biological characteristics. They are also common in chiral ligands used for asymmetric syntheses and as synthetic intermediates. Herein, we present asymmetric routes to 2,4,5-trisubstituted Δ(2)-thiazolines. These Δ(2)-thiazolines were synthesized from readily accessible/commercially available α,β-unsaturated methyl es...

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ژورنال

عنوان ژورنال: Chemistry - A European Journal

سال: 2013

ISSN: 0947-6539

DOI: 10.1002/chem.201301120