Intestinal permeability and transport of apigenin across caco-2 cell monolayers
نویسندگان
چکیده
منابع مشابه
Transport characteristics of ebastine and its metabolites across human intestinal epithelial Caco-2 cell monolayers.
The transport characteristics of a selective peripheral H1 receptor antagonist, ebastine, a substrate for cytochrome P450 3A4, and its three major metabolites, i.e., the hydroxy metabolite of ebastine (M-OH), the pharmacologically active metabolite carebastine (Car), and the desbutyrophenone metabolite (des-BP), were studied in cultured human intestinal Caco-2 cells expressing a drug efflux pum...
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Although being reported and used as a sedative remedy for several years, the bioactive principle of hop preparations is still not decisively clarified. Understanding absorption and transformation processes of potential physiologically active constituents is essential to evaluate the likeliness of biological effects on humans. Therefore, single hop aroma compounds as well as digestive transforma...
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ژورنال
عنوان ژورنال: Journal of Food Bioactives
سال: 2019
ISSN: 2637-8779,2637-8752
DOI: 10.31665/jfb.2019.7198