Ligand efficiency as a guide in fragment hit selection and optimization
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چکیده
منابع مشابه
Ligand efficiency as a guide in fragment hit selection and optimization.
Ligand efficiency as a guide in fragment hit selection and optimization Sabine Schultes, Chris de Graaf, Eric E.J. Haaksma*, Iwan J.P. de Esch, Rob Leurs, Oliver Krämer Boehringer Ingelheim RCV GmbH & Co. KG, Department of Medicinal Chemistry, Dr. Boehringer-Gasse 5-11, Vienna, Austria Leiden/Amsterdam Center for Drug Research (LACDR), Division of Medicinal Chemistry, Department of Pharmacochem...
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ژورنال
عنوان ژورنال: Drug Discovery Today: Technologies
سال: 2010
ISSN: 1740-6749
DOI: 10.1016/j.ddtec.2010.11.003