نتایج جستجو برای: benzyl thio

تعداد نتایج: 12199  

A novel series of azolylalkylthio, -sulfoxy, and-sulfonyl compounds was designed, synthesized, and evaluated for antipicornaviral activity. Two compounds (4i and 4 1) exhibited significant activity against various serotypes of human rhinovirus (HRV). It was found that incorporation of hydrophobic azoles such as 3-methylisoxazole or 4-methylthiazole led to increased activity. In addition, ac...

2013
Larissa Leffers Christoph A. Wehe Sabine Hüwel Marc Bartel Franziska Ebert Mojtaba S. Taleshi Hans-Joachim Galla Uwe Karst Kevin A. Francesconi Tanja Schwerdtle

Whereas inorganic arsenic is classified as a human carcinogen, risks to human health related to the presence of arsenosugars in marine food are still unclear. Since studies indicate that human inorganic arsenic metabolites contribute to inorganic arsenic induced carcinogenicity, a risk assessment for arsenosugars should also include a toxicological characterization of their respective metabolit...

2017
Elizabeth Leese Malcolm Clench Jackie Morton Philip H E Gardiner Vikki A Carolan

This study investigates the identity of two unexpected arsenic species found separately in a number of urine samples sent to the Health and Safety Executive's Health and Safety Laboratory for arsenic speciation (arsenobetaine, AB; arsenite, As3+; arsenate, As5+; monomethylarsonic acid, MMA5+; and dimethylarsinic acid, DMA5+). Micro liquid chromatography coupled to inductively coupled plasma mas...

2017
Kyoung Mi Moon Bonggi Lee Ji Won Jeong Dae Hyun Kim Yun Jung Park Hye Rim Kim Ji Young Park Min Jo Kim Hye Jin An Eun Kyeong Lee Young Mi Ha Eunok Im Pusoon Chun Jin Yeul Ma Won-Kyung Cho Hyung Ryong Moon Hae Young Chung

Liver inflammation is closely associated with metabolic syndrome. Oxidative stress plays a synergistic role in inflammation by activating nuclear factor kappa B (NF-κB) signaling in the liver. Therefore, substantial efforts have been made to develop compounds that inhibit the generation of oxidative stress and activation of NF-κB. We synthesized twenty-six novel 5-(substituted benzyl)-2-oxo- an...

Journal: :Molecular pharmacology 2003
Annamaria De Luca Sophie Talon Michela De Bellis Jean-François Desaphy Giovanni Lentini Filomena Corbo Antonio Scilimati Carlo Franchini Vincenzo Tortorella Diana Conte Camerino

Newly synthesized tocainide analogs were tested for their state-dependent affinity and use-dependent behavior on sodium currents (INa) of adult skeletal muscle fibers by means of the Vaseline-gap voltage clamp method. The drugs had the pharmacophore amino group constrained in position alpha [N-(2,6-dimethylphenyl)pyrrolidine-2-carboxamide (To5)] or beta [N-(2,6-dimethylphenyl)pyrrolidine-3-carb...

BiFeO3 (BFO), Bi0.86Sm0.07Eu0.07FeO3 (BSEFO), and Bi0.86Sm0.07Cd0.07FeO3 (BSCFO) nano powders were prepared by the sol-gel combustion method and the catalytic performances were evaluated in the acetylation reaction of benzyl alcohol. The physical chemical properties of the catalysts were character...

In this study, TiO2-10%wt. carbon nanotube (CNT) nanocomposite powders were synthesized by sol-gel method at various hydrolysis rate affected by different reaction agents of acetyl acetone and benzyl alcohol. Crystallization of TiO2 was then achieved through calcination at 400 °C. The properties of nanocomposite powder investigated by scanning electron microscopy, X-ray diffraction and diffuse ...

Journal: :journal of sciences islamic republic of iran 0

a novel series of azolylalkylthio, -sulfoxy, and-sulfonyl compounds was designed, synthesized, and evaluated for antipicornaviral activity. two compounds (4i and 4 1) exhibited significant activity against various serotypes of human rhinovirus (hrv). it was found that incorporation of hydrophobic azoles such as 3-methylisoxazole or 4-methylthiazole led to increased activity. in addition, activi...

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